SCHEMBL30848845

SCHEMBL30848845

O=S(=O)(Oc1ccc(Br)c2cnc(Cl)cc12)C(F)(F)F

nearest known ligand 0.34

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
EPAS1 Q99814 7/20 0.34
CSNK2A1 P68400 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.32
PDE4A P27815 1/20 0.32
PDE4C Q08493 1/20 0.32
PDE4D Q08499 1/20 0.32
ESR2 Q92731 1/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
ALPL P05186 2/20 0.31
ADORA2A P29274 1/20 0.30
ADORA1 P30542 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23579175 1.00 EPAS1 (0.34) EPAS1CSNK2A1L3MBTL1PDE4APDE4C
SCHEMBL30150671 1.00 EPAS1 (0.34) EPAS1CSNK2A1L3MBTL1PDE4APDE4C
SCHEMBL29206714 0.82 CSNK2A1 (0.35) EPAS1CSNK2A1ALPL
SCHEMBL29959365 0.80 CSNK2A1 (0.32) CSNK2A1PDE4APDE4CPDE4D
SCHEMBL23578707 0.80 CSNK2A1 (0.32) CSNK2A1PDE4APDE4CPDE4D
SCHEMBL2185158 0.77 PDE4A (0.34) PDE4APDE4CPDE4DESR2CA1
SCHEMBL24819988 0.77 L3MBTL1 (0.34) CSNK2A1L3MBTL1
SCHEMBL23592754 0.74 NQO1 (0.39) CSNK2A1
SCHEMBL21313423 0.74 PKM (0.43) EPAS1L3MBTL1ESR2CA1CA2
SCHEMBL1396954 0.74 PDE4A (0.36) EPAS1L3MBTL1PDE4APDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250368616-A1 NITROGEN-CONTAINING HETEROCYCLIC DERIVATIVE INHIBITOR, AND PREPARATION METHOD THEREFOR AND USE THEREOF SHANGHAI HANSOH BIOMEDICAL CO LTD (CN) 2025-12-04 US disclosed
US-20250206718-A1 NITROGEN-CONTAINING HETEROCYCLIC DERIVATIVE INHIBITOR, PREPARATION METHOD THEREFOR AND USE THEREOF JIANGSU HANSOH PHARMACEUTICAL GROUP CO., LTD. (CN) 2025-06-26 US disclosed
EP-4495110-A1 NITROGEN-CONTAINING HETEROCYCLIC DERIVATIVE INHIBITOR, PREPARATION METHOD THEREFOR AND USE THEREOF Shanghai Hansoh Biomedical Co., Ltd. (CN) 2025-01-22 EP disclosed
CN-118871433-A Nitrogen-containing heterocyclic derivative inhibitor, preparation method and application thereof 上海翰森生物医药科技有限公司 2024-10-29 CN disclosed
CN-117940424-A EGFR inhibitors 缆图药品公司 2024-04-26 CN disclosed
CN-117916232-A Heterocyclic EGFR inhibitors for the treatment of cancer 缆图药品公司 2024-04-19 CN disclosed
CN-117858872-A Heterocyclic EGFR inhibitors for the treatment of cancer 缆图药品公司 2024-04-09 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250206718-A1 NITROGEN-CONTAINING HETEROCYCLIC DERIVATIVE INHIBITOR, PREPARATION METHOD THEREFOR AND USE THEREOF WEE1, EGFR, WEE2 EPAS1 2594/4885CSNK2A1 1381/4885L3MBTL1 4742/4885
US-20250368616-A1 NITROGEN-CONTAINING HETEROCYCLIC DERIVATIVE INHIBITOR, AND PREPARATION METHOD THEREFOR AND USE THEREOF WEE1, WEE2, EGFR EPAS1 2252/4885CSNK2A1 2155/4885L3MBTL1 4118/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.