SCHEMBL30849541

SCHEMBL30849541

[2H]c1ncnc2[nH]cc(C#C)c12

nearest known ligand 0.33

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 1/20 0.33
AAK1 Q2M2I8 1/20 0.33
RPS6KA5 O75582 1/20 0.31
DPYD Q12882 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1799199 0.82 RPS6KA5 (0.42) LRRK2AAK1RPS6KA5DPYD
SCHEMBL25839045 0.66 AAK1 (0.38) LRRK2AAK1DPYD
SCHEMBL5522171 0.64 LRRK2 (0.40) LRRK2DPYD
SCHEMBL5260963 0.64 LRRK2 (0.54) LRRK2AAK1RPS6KA5
SCHEMBL30199352 0.64 LRRK2 (0.54) LRRK2AAK1RPS6KA5
SCHEMBL9254230 0.63 JAK3 (0.39) LRRK2DPYD
SCHEMBL1737697 0.63 CHEK1 (0.56) LRRK2DPYD
Hydrochloric Acid SCHEMBL28274256 0.63 LRRK2 (0.53) LRRK2AAK1RPS6KA5
SCHEMBL30849544 0.63 CDK8 (0.53) RPS6KA5
Purine SCHEMBL30151982 0.58

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117460736-A Nucleoside derivatives having multi-target phosphorylase inhibitory activity and pharmaceutical compositions for preventing and treating cancer comprising the same 未来制药有限公司 2024-01-26 CN disclosed