SCHEMBL9254230

SCHEMBL9254230

C#Cc1c[nH]c2ncnc(O)c12

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
JAK3 P52333 1/20 0.39
MAP3K7 O43318 3/20 0.36
TAB1 Q15750 3/20 0.36
CHEK1 O14757 1/20 0.36
CHUK O15111 2/20 0.34
HSP90AB1 P08238 1/20 0.34
AKT1 P31749 3/20 0.33
LRRK2 Q5S007 4/20 0.33
IRAK4 Q9NWZ3 1/20 0.32
DPYD Q12882 1/20 0.32
NOTUM Q6P988 1/20 0.31
ROCK2 O75116 2/20 0.31
ROCK1 Q13464 2/20 0.31
CDC42BPA Q5VT25 2/20 0.31
CDC42BPB Q9Y5S2 2/20 0.31
IKBKB O14920 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1737697 0.79 CHEK1 (0.56) JAK3MAP3K7TAB1CHEK1CHUK
SCHEMBL7885565 0.72 MAPK1 (0.39) JAK3MAP3K7TAB1CHEK1CHUK
SCHEMBL7887899 0.72 CHEK1 (0.61) JAK3MAP3K7TAB1CHEK1CHUK
SCHEMBL15618411 0.68 IRAK4 (0.47) MAP3K7TAB1CHEK1LRRK2IRAK4
SCHEMBL30975034 0.68 IRAK4 (0.47) JAK3MAP3K7TAB1CHEK1LRRK2
SCHEMBL1806375 0.65 MAP3K7 (0.41) JAK3MAP3K7TAB1CHEK1NOTUM
SCHEMBL30849541 0.63 LRRK2 (0.33) LRRK2DPYD
SCHEMBL14649086 0.61 MAP3K7 (0.56) MAP3K7TAB1CHUKHSP90AB1LRRK2
SCHEMBL12590787 0.60 CHUK (0.48) JAK3MAP3K7TAB1CHUKHSP90AB1
SCHEMBL31612016 0.59 CDC7 (0.50) JAK3MAP3K7TAB1CHEK1CHUK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5426187-A Process for the preparation of 4-hydroxy-5-substituted ethynylpyrrolo [2,3-d]pyrimidine intermediates ELI LILLY AND COMPANY (US) 1995-06-20 US disclosed