SCHEMBL3085107

SCHEMBL3085107

O=C(O)n1c(=O)[nH]c2nc[nH]c2c1=O

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 7/20 0.58
ADORA2A P29274 4/20 0.58
PDE4A P27815 3/20 0.54
PDE4B Q07343 3/20 0.54
PDE4C Q08493 3/20 0.54
PDE4D Q08499 3/20 0.54
ADORA3 P0DMS8 6/20 0.51
GDA Q9Y2T3 2/20 0.43
ACHE P22303 1/20 0.43
ABL1 P00519 1/20 0.40
RIN1 Q13671 1/20 0.40
ADORA1 P30542 1/20 0.37
TDP1 Q9NUW8 2/20 0.36
ALDH1A1 P00352 2/20 0.35
KDM4E B2RXH2 1/20 0.35
TP53 P04637 1/20 0.35
HPGD P15428 1/20 0.35
PTGS1 P23219 1/20 0.35
HBB P68871 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6555067 0.85 ADORA2B (0.57) ADORA2BADORA2APDE4APDE4BPDE4C
SCHEMBL8884694 0.85 ADORA2B (0.61) ADORA2BADORA2APDE4APDE4BPDE4C
SCHEMBL7491449 0.81 ADORA2B (0.56) ADORA2BADORA2APDE4APDE4BPDE4C
SCHEMBL7800909 0.79 ADORA2B (0.50) ADORA2BADORA2APDE4APDE4BPDE4C
SCHEMBL618977 0.77 ADORA2B (0.64) ADORA2BADORA2APDE4APDE4BPDE4C
SCHEMBL18285098 0.77 ADORA2A (0.55) ADORA2BADORA2APDE4APDE4BPDE4C
SCHEMBL8952223 0.77 ADORA2A (0.55) ADORA2BADORA2APDE4APDE4BPDE4C
SCHEMBL11572222 0.76 ADORA2B (0.59) ADORA2BADORA2APDE4APDE4BPDE4C
Hydrochloric Acid SCHEMBL28403443 0.76 ADORA2B (0.62) ADORA2BADORA2APDE4APDE4BPDE4C
1-Methylxanthine SCHEMBL7270651 0.74 ADORA2B (0.77) ADORA2BADORA2APDE4APDE4BPDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 56 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20180055868-A1 METHODS AND COMPOSITIONS FOR STIMULATING BONE REGENERATION NEW YORK UNIVERSITY (US) 2018-03-01 US disclosed
US-20160262894-A1 TISSUE REPAIR DEVICES AND SCAFFOLDS NATIONAL INSTITUTES OF HEALTH - DIRECTOR DEITR 2016-09-15 US disclosed
WO-2015065819-A1 TISSUE REPAIR DEVICES AND SCAFFOLDS NEW YORK UNIVERSITY (US) 2015-05-07 WO disclosed
US-20150011496-A1 METHODS AND COMPOSITIONS FOR STIMULATING BONE REGENERATION NEW YORK UNIVERSITY 2015-01-08 US disclosed
WO-2013126545-A1 METHODS AND COMPOSITIONS FOR STIMULATING BONE REGENERATION NEW YORK UNIVERSITY (US) 2013-08-29 WO disclosed
US-7795427-B2 Methods for inhibiting osteoclast differentiation, formation, or function and for increasing bone mass NEW YORK UNIVERSITY (US) 2010-09-14 US disclosed
US-7335655-B2 8-heteroaryl xanthine adenosine A2B receptor antagonists KING PHARMACEUTICALS RESEARCH AND DEVELOPMENT, INC. (US) 2008-02-26 US disclosed
WO-2007095161-A2 METHODS AND COMPOSITIONS FOR TREATING DISORDERS ASSOCIATED WITH INCREASED BONE TURNOVER AND OSTEOPENIA NEW YORK UNIVERSITY (US) 2007-08-23 WO disclosed
US-20070191279-A1 Methods and compositions for treating disorders associated with increased bone turnover and osteopenia CRONSTEIN BRUCE N 2007-08-16 US disclosed
US-7205403-B2 8-Heteroaryl xanthine adenosine A2B receptor antagonists KING PHARMACEUTICALS RESEARCH AND DEVELOPMENT, INC. (US) 2007-04-17 US disclosed
US-5733916-A RESPIRATORY SYSTEM DISORDERS THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 1998-03-31 US disclosed
EP-0793406-A1 Process for producing multilayer wiring boards TOKYO OHKA KOGYO CO., LTD. (JP) 1997-09-03 EP disclosed
EP-0755254-A1 PREVENTION AND TREATMENT OF ISCHEMIA-REPERFUSION AND ENDOTOXIN-RELATED INJURY USING ADENOSINE AND PURINO RECEPTOR ANTAGONISTS THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 1997-01-29 EP disclosed
US-5504090-A Compositions and methods for the prevention and treatment of ischemia-reperfusion organ injury TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 1996-04-02 US disclosed
WO-1995026728-A1 PREVENTION AND TREATMENT OF ISCHEMIA-REPERFUSION AND ENDOTOXIN-RELATED INJURY USING ADENOSINE AND PURINO RECEPTOR ANTAGONISTS THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 1995-10-12 WO disclosed
US-5453426-A Sulfur-containing xanthine derivatives as adenosine antagonists THE UNITED STATES OF AMERICA AS REPRESENTED BY THE DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 1995-09-26 US disclosed
US-4968672-A DRUG DELIVERY; DIURETICS, KIDNEY DISORDERS, HYPOTENSIVE AGENTS THE UNITED STATES OF AMERICA AS REPRESENTED BY THE DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 1990-11-06 US disclosed
WO-1990012797-A1 SULFER-CONTAINING XANTHINE DERIVATIVES AS ADENOSIN ANTAGONISTS THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, U.S. DEPARTMENT OF COMMERCE (US) 1990-11-01 WO disclosed
US-4741818-A COMPLEXES LEARONAL, INC. (US) 1988-05-03 US disclosed
EP-0225422-A1 Alkaline baths and methods for electrodeposition of palladium and palladium alloys LeaRonal, Inc. (US) 1987-06-16 EP disclosed