1-Methylxanthine

1-Methylxanthine

SCHEMBL7270651

CCC(=O)O.Cn1c(=O)[nH]c2nc[nH]c2c1=O

nearest known ligand 0.77

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 10/20 0.77
ADORA2A P29274 8/20 0.77
ADORA3 P0DMS8 7/20 0.59
PDE4A P27815 7/20 0.59
PDE4B Q07343 7/20 0.59
PDE4C Q08493 7/20 0.59
PDE4D Q08499 7/20 0.59
ATAD2 Q6PL18 1/20 0.42
PIK3CD O00329 1/20 0.41
ALPL P05186 1/20 0.41
TMIGD3 P0DMS9 1/20 0.41
ADORA1 P30542 1/20 0.41
CYP2C19 P33261 1/20 0.41
HIF1A Q16665 1/20 0.41
ALDH1A1 P00352 1/20 0.41
LMNA P02545 1/20 0.41
CYP3A4 P08684 1/20 0.41
MAPT P10636 1/20 0.41
TSHR P16473 1/20 0.41
BLM P54132 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
1-Methylxanthine SCHEMBL10996 0.88 ADORA2B (1.00) ADORA2BADORA2AADORA3PDE4APDE4B
1-Methylxanthine SCHEMBL27529726 0.86 ADORA2B (0.96) ADORA2BADORA2AADORA3PDE4APDE4B
1-Methylxanthine SCHEMBL9682658 0.86 ADORA2B (0.96) ADORA2BADORA2AADORA3PDE4APDE4B
1-Methylxanthine SCHEMBL28309011 0.86 ADORA2B (0.96) ADORA2BADORA2AADORA3PDE4APDE4B
1-Methylxanthine SCHEMBL28460409 0.84 ADORA2B (0.84) ADORA2BADORA2AADORA3PDE4APDE4B
1-Methylxanthine SCHEMBL27663813 0.83 ADORA2B (0.77) ADORA2BADORA2AADORA3PDE4APDE4B
1-Methylxanthine SCHEMBL17748264 0.82 ADORA2B (0.89) ADORA2BADORA2AADORA3PDE4APDE4B
1-Methylxanthine SCHEMBL29001829 0.81 ADORA2B (0.79) ADORA2BADORA2AADORA3PDE4APDE4B
1-Methylxanthine SCHEMBL16859909 0.78 ADORA2B (0.79) ADORA2BADORA2AADORA3PDE4APDE4B
Theophylline Anhydrous SCHEMBL1128138 0.77 ADORA2A (0.77) ADORA2BADORA2AADORA3PDE4APDE4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20030186339-A1 Individualization of therapy with antibiotic agents MCGILL UNIVERSITY 2003-10-02 US disclosed