SCHEMBL30853060

SCHEMBL30853060

C[C@@H]1CCOc2nccc(NC(=O)OC(C)(C)C)c2O1

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
METAP1 P53582 1/20 0.38
ATR Q13535 1/20 0.37
BRS3 P32247 1/20 0.34
BRAF P15056 1/20 0.34
NPSR1 Q6W5P4 1/20 0.32
ACACB O00763 1/20 0.32
ACACA Q13085 1/20 0.32
BRD9 Q9H8M2 1/20 0.32
CYP17A1 P05093 2/20 0.32
DGAT1 O75907 1/20 0.32
GSK3B P49841 1/20 0.32
DYRK1A Q13627 1/20 0.32
KDM4D Q6B0I6 1/20 0.32
RORC P51449 1/20 0.32
CHRM1 P11229 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24752319 1.00 METAP1 (0.38) METAP1ATRBRS3BRAFNPSR1
SCHEMBL3198182 0.80 ATR (0.41) METAP1ATRBRD9CYP17A1
SCHEMBL3588883 0.72 KCNH2 (0.43) KDM4D
SCHEMBL29127965 0.69 RORC (0.41) METAP1ATRBRS3BRAFACACB
SCHEMBL34466677 0.66 ATR (0.38) METAP1ATRBRS3CYP17A1CHRM1
SCHEMBL31570618 0.65 GAA (0.40) METAP1ATRBRS3BRAFCYP17A1
SCHEMBL31570445 0.65 ATR (0.42) METAP1ATRBRS3BRAFACACB
SCHEMBL30888170 0.65 ATR (0.59) METAP1ATRCYP17A1
SCHEMBL16992920 0.65 ATR (0.46) METAP1ATRBRD9CYP17A1
SCHEMBL7949833 0.65 MRGPRX1 (0.46) BRD9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117881681-A Substituted pyrrolo [2,3-d ] pyrimidines, their preparation and their therapeutic use 赛诺菲 2024-04-12 CN disclosed