SCHEMBL30853474

SCHEMBL30853474

CCOC(=O)c1cc2cccnc2c(=O)[nH]1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 4/20 0.54
KDM4E B2RXH2 4/20 0.54
ALDH1A1 P00352 4/20 0.54
HPGD P15428 4/20 0.54
LMNA P02545 3/20 0.54
SMN1; SMN2 Q16637 2/20 0.54
NPC1 O15118 2/20 0.54
MAPT P10636 2/20 0.54
MEN1 O00255 1/20 0.54
GLA P06280 1/20 0.54
GAA P10253 1/20 0.54
KMT2A Q03164 1/20 0.54
ATM Q13315 1/20 0.54
MMP13 P45452 7/20 0.53
MMP2 P08253 5/20 0.53
MMP14 P50281 3/20 0.53
HSD17B10 Q99714 2/20 0.52
POLB P06746 2/20 0.51
HTT P42858 2/20 0.49
L3MBTL1 Q9Y468 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16505827 1.00 RAB9A (0.54) RAB9AKDM4EALDH1A1HPGDLMNA
SCHEMBL832252 0.82 KDM4E (0.58) RAB9AKDM4EALDH1A1HPGDLMNA
SCHEMBL30023186 0.79 HSD17B10 (0.49) KDM4EALDH1A1HPGDLMNASMN1; SMN2
SCHEMBL22411420 0.78 CYP1A2 (0.50) RAB9AKDM4EALDH1A1HPGDLMNA
SCHEMBL30873871 0.78 CYP1A2 (0.50) RAB9AKDM4EALDH1A1HPGDLMNA
SCHEMBL15367087 0.78 KDM4E (0.63) RAB9AKDM4EALDH1A1HPGDLMNA
SCHEMBL16008122 0.76 CDK1 (0.57) RAB9AKDM4EALDH1A1HPGDLMNA
SCHEMBL13064936 0.76 ALDH1A1 (0.57) RAB9AKDM4EALDH1A1HPGDLMNA
SCHEMBL16505498 0.75 CYP1A2 (0.49) RAB9AKDM4EALDH1A1HPGDNPC1
SCHEMBL22428818 0.75 PDE4A (0.52) KDM4EALDH1A1HPGDSMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4524136-A1 KINESIN KIF18A INHIBITOR AND USE THEREOF Shanghai Apeiron Therapeutics Company Limited (CN) 2025-03-19 EP disclosed
CN-119156382-A Kinesin KIF18A inhibitor and application thereof 上海湃隆生物科技有限公司 2024-12-17 CN disclosed
CN-115397822-B CBP/EP300 inhibitors and uses thereof 南京药石科技股份有限公司 2024-04-16 CN disclosed