SCHEMBL30853520

SCHEMBL30853520

NC(=O)c1ccc(-n2ccc3c(Nc4ccc(C(F)(F)F)cc4)ncnc32)cc1NC1CCCCC1

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PIP4K2A P48426 3/20 0.45
PIK3CG P48736 3/20 0.45
SOS1 Q07889 1/20 0.43
RPS6KB1 P23443 2/20 0.41
PDPK1 O15530 1/20 0.41
HSP90AA1 P07900 2/20 0.41
JAK2 O60674 3/20 0.41
JAK1 P23458 3/20 0.41
TRPV1 Q8NER1 1/20 0.41
EGFR P00533 3/20 0.40
FLT3 P36888 1/20 0.40
ERBB2 P04626 1/20 0.39
AURKA O14965 1/20 0.39
AURKB Q96GD4 1/20 0.39
PAK1 Q13153 1/20 0.39
SYK P43405 2/20 0.38
ABL1 P00519 1/20 0.38
BCR P11274 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30853530 0.93 HSP90AA1 (0.49) PIP4K2APIK3CGHSP90AA1JAK2JAK1
SCHEMBL30853531 0.92 PIP4K2A (0.47) PIP4K2APIK3CGSOS1HSP90AA1TRPV1
SCHEMBL30853526 0.89 PIP4K2A (0.46) PIP4K2APIK3CGHSP90AA1JAK2SYK
SCHEMBL30853539 0.87 PIP4K2A (0.47) PIP4K2APIK3CGHSP90AA1SYK
SCHEMBL30853536 0.86 PIP4K2A (0.45) PIP4K2APIK3CGSOS1HSP90AA1SYK
SCHEMBL30853533 0.86 PIP4K2A (0.46) PIP4K2APIK3CGHSP90AA1EGFRERBB2
SCHEMBL30853529 0.84 PIP4K2A (0.51) PIP4K2APIK3CGRPS6KB1HSP90AA1AURKB
SCHEMBL30853521 0.84 CTSS (0.43) PIP4K2APIK3CGSOS1JAK2TRPV1
SCHEMBL30853542 0.82 HSP90AA1 (0.54) PIP4K2APIK3CGHSP90AA1
SCHEMBL30853519 0.81 HSP90AA1 (0.43) PIP4K2APIK3CGHSP90AA1JAK2JAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118047781-A HSP90 inhibitor and preparation method and application thereof 广西大学 2024-05-17 CN disclosed