SCHEMBL30853832

SCHEMBL30853832

Nc1cccc(-c2nncn2C2CCC2)c1

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MAP3K5 Q99683 7/20 0.45
KDM4E B2RXH2 1/20 0.44
HPGD P15428 2/20 0.41
ALDH1A1 P00352 1/20 0.41
HSD17B10 Q99714 1/20 0.41
MAP4K1 Q92918 4/20 0.38
TNF P01375 2/20 0.36
ABL1 P00519 1/20 0.36
EGFR P00533 1/20 0.36
SRC P12931 1/20 0.36
ABL2 P42684 1/20 0.36
MAOA P21397 1/20 0.36
MYLK Q15746 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL944155 0.94 MAP3K5 (0.43) MAP3K5KDM4EHPGDALDH1A1HSD17B10
SCHEMBL30853796 0.94 MAP3K5 (0.43) MAP3K5KDM4EHPGDALDH1A1HSD17B10
SCHEMBL857728 0.75 ALDH1A1 (0.43) KDM4EHPGDALDH1A1HSD17B10MAOA
SCHEMBL22126011 0.75 TNF (0.38) MAP3K5ALDH1A1TNFMYLK
SCHEMBL20802751 0.74 MAP3K5 (0.48) MAP3K5MAP4K1TNFMYLK
SCHEMBL6127726 0.74 MAP3K5 (0.48) MAP3K5TNFMYLK
SCHEMBL28987781 0.73 MAP3K5 (0.42) MAP3K5MAP4K1TNFEGFRMYLK
SCHEMBL20802774 0.71 MAP3K5 (0.48) MAP3K5MAP4K1TNFMYLK
SCHEMBL29664258 0.71 MAP4K4 (0.41) KDM4EHPGDALDH1A1HSD17B10SRC
SCHEMBL22404532 0.70 MAP3K5 (0.47) MAP3K5MAP4K1TNFMYLK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117903128-A ASK1/PDK1 double-targeting inhibitor, and preparation method and application thereof 中南大学 2024-04-19 CN disclosed