SCHEMBL30878397

SCHEMBL30878397

C#Cc1c(-c2ccccc2Cl)c(=O)n(C)c2nc(Nc3ccccc3OC)ncc12

nearest known ligand 0.64

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
EGFR P00533 7/20 0.64
FGFR1 P11362 7/20 0.64
WEE1 P30291 6/20 0.57
IGF1R P08069 5/20 0.52
LRRK2 Q5S007 1/20 0.47
LCK P06239 1/20 0.46
PTK2 Q05397 1/20 0.46
SRC P12931 2/20 0.45
FGFR2 P21802 1/20 0.44
FGFR4 P22455 1/20 0.44
FGFR3 P22607 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30878805 0.88 EGFR (0.56) EGFRFGFR1WEE1IGF1RLRRK2
SCHEMBL30878354 0.86 IGF1R (0.60) EGFRIGF1RLRRK2PTK2SRC
SCHEMBL30878366 0.85 FGFR1 (0.66) EGFRFGFR1WEE1SRCFGFR2
SCHEMBL30878465 0.85 WEE1 (0.77) EGFRFGFR1WEE1SRCFGFR2
SCHEMBL30878347 0.85 EGFR (0.61) EGFRFGFR1WEE1IGF1RLRRK2
SCHEMBL30878436 0.85 EGFR (0.49) EGFRFGFR1WEE1IGF1RLRRK2
SCHEMBL30878328 0.80 EGFR (0.50) EGFRFGFR1WEE1IGF1RLRRK2
SCHEMBL30878310 0.79 EGFR (0.65) EGFRFGFR1WEE1IGF1RLRRK2
SCHEMBL30878321 0.78 EGFR (0.54) EGFRFGFR1WEE1IGF1RLRRK2
SCHEMBL5762573 0.78 FGFR1 (1.00) EGFRFGFR1WEE1SRCFGFR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4612148-A1 2-AMINO-PYRIDO[2,3-D]PYRIMIDIN-7(8H)-ONE AND 7-AMINO-1-PYRIMIDO[4,5-D]PYRIMIDIN-2(1 H)-ONE DERIVATIVES AS EGFR INHIBITORS FOR THE TREATMENT OF CANCER Cancer Research Technology Limited (GB) 2025-09-10 EP claimed
WO-2024094963-A1 2-AMINO-PYRIDO[2,3-D]PYRIMIDIN-7(8H)-ONE AND 7-AMINO-1-PYRIMIDO[4,5-D]PYRIMIDIN-2(1 H)-ONE DERIVATIVES AS EGFR INHIBITORS FOR THE TREATMENT OF CANCER CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2024-05-10 WO claimed
EP-4612148-A1 2-AMINO-PYRIDO[2,3-D]PYRIMIDIN-7(8H)-ONE AND 7-AMINO-1-PYRIMIDO[4,5-D]PYRIMIDIN-2(1 H)-ONE DERIVATIVES AS EGFR INHIBITORS FOR THE TREATMENT OF CANCER Cancer Research Technology Limited (GB) 2025-09-10 EP disclosed
WO-2024094963-A1 2-AMINO-PYRIDO[2,3-D]PYRIMIDIN-7(8H)-ONE AND 7-AMINO-1-PYRIMIDO[4,5-D]PYRIMIDIN-2(1 H)-ONE DERIVATIVES AS EGFR INHIBITORS FOR THE TREATMENT OF CANCER CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2024-05-10 WO disclosed