SCHEMBL30878436

SCHEMBL30878436

C#Cc1c(-c2ccccc2Cl)c(=O)n(C)c2nc(Nc3ccc(N(C)CCN(C)C)cc3OC)ncc12

nearest known ligand 0.49

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
EGFR P00533 9/20 0.49
FGFR1 P11362 6/20 0.49
BTK Q06187 2/20 0.47
JAK3 P52333 1/20 0.46
WEE1 P30291 3/20 0.46
IGF1R P08069 4/20 0.44
MAPK7 Q13164 1/20 0.42
LRRK2 Q5S007 1/20 0.42
SRC P12931 2/20 0.41
TNK2 Q07912 1/20 0.41
KCNH2 Q12809 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30879162 0.90 EGFR (0.48) EGFRFGFR1BTKJAK3WEE1
SCHEMBL30878362 0.90 EGFR (0.49) EGFRFGFR1BTKJAK3WEE1
SCHEMBL30878325 0.86 WEE1 (0.58) EGFRFGFR1WEE1SRCTNK2
SCHEMBL30878313 0.85 EGFR (0.49) EGFRFGFR1BTKJAK3MAPK7
SCHEMBL30878397 0.85 EGFR (0.64) EGFRFGFR1WEE1IGF1RLRRK2
SCHEMBL30878353 0.84 FGFR4 (0.47) EGFRFGFR1BTKWEE1SRC
SCHEMBL30878454 0.83 FGFR1 (0.51) EGFRFGFR1BTKJAK3WEE1
SCHEMBL30878484 0.82 EGFR (0.52) EGFRBTKJAK3MAPK7LRRK2
SCHEMBL30878354 0.81 IGF1R (0.60) EGFRIGF1RMAPK7LRRK2SRC
SCHEMBL30878727 0.80 EGFR (0.50) EGFRFGFR1BTKJAK3IGF1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4612148-A1 2-AMINO-PYRIDO[2,3-D]PYRIMIDIN-7(8H)-ONE AND 7-AMINO-1-PYRIMIDO[4,5-D]PYRIMIDIN-2(1 H)-ONE DERIVATIVES AS EGFR INHIBITORS FOR THE TREATMENT OF CANCER Cancer Research Technology Limited (GB) 2025-09-10 EP claimed
WO-2024094963-A1 2-AMINO-PYRIDO[2,3-D]PYRIMIDIN-7(8H)-ONE AND 7-AMINO-1-PYRIMIDO[4,5-D]PYRIMIDIN-2(1 H)-ONE DERIVATIVES AS EGFR INHIBITORS FOR THE TREATMENT OF CANCER CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2024-05-10 WO claimed
EP-4612148-A1 2-AMINO-PYRIDO[2,3-D]PYRIMIDIN-7(8H)-ONE AND 7-AMINO-1-PYRIMIDO[4,5-D]PYRIMIDIN-2(1 H)-ONE DERIVATIVES AS EGFR INHIBITORS FOR THE TREATMENT OF CANCER Cancer Research Technology Limited (GB) 2025-09-10 EP disclosed
WO-2024094963-A1 2-AMINO-PYRIDO[2,3-D]PYRIMIDIN-7(8H)-ONE AND 7-AMINO-1-PYRIMIDO[4,5-D]PYRIMIDIN-2(1 H)-ONE DERIVATIVES AS EGFR INHIBITORS FOR THE TREATMENT OF CANCER CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2024-05-10 WO disclosed