SCHEMBL30878347

SCHEMBL30878347

C=Cc1c(-c2ccccc2Cl)c(=O)n(C)c2nc(Nc3ccccc3OC)ncc12

nearest known ligand 0.61

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
EGFR P00533 7/20 0.61
FGFR1 P11362 7/20 0.61
WEE1 P30291 3/20 0.55
IGF1R P08069 3/20 0.49
LRRK2 Q5S007 1/20 0.48
BTK Q06187 1/20 0.47
ALK Q9UM73 2/20 0.45
LCK P06239 1/20 0.45
JAK3 P52333 1/20 0.44
PTK2 Q05397 1/20 0.44
SRC P12931 1/20 0.44
INSR P06213 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30878310 0.92 EGFR (0.65) EGFRFGFR1WEE1IGF1RLRRK2
SCHEMBL30878488 0.87 EGFR (0.53) EGFRFGFR1WEE1IGF1RLRRK2
SCHEMBL30878322 0.87 EGFR (0.59) EGFRIGF1RLRRK2ALKPTK2
SCHEMBL30878358 0.86 FGFR1 (0.64) EGFRFGFR1WEE1SRC
SCHEMBL30878397 0.85 EGFR (0.64) EGFRFGFR1WEE1IGF1RLRRK2
SCHEMBL30878805 0.79 EGFR (0.56) EGFRFGFR1WEE1IGF1RLRRK2
SCHEMBL30878501 0.78 FGFR1 (0.53) EGFRFGFR1WEE1SRC
SCHEMBL30878459 0.78 ABL1 (0.65) EGFRFGFR1WEE1SRC
SCHEMBL30878475 0.78 SRC (0.63) FGFR1WEE1ALKLCKSRC
SCHEMBL30878382 0.78 WEE1 (0.70) EGFRFGFR1WEE1IGF1RLRRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4612148-A1 2-AMINO-PYRIDO[2,3-D]PYRIMIDIN-7(8H)-ONE AND 7-AMINO-1-PYRIMIDO[4,5-D]PYRIMIDIN-2(1 H)-ONE DERIVATIVES AS EGFR INHIBITORS FOR THE TREATMENT OF CANCER Cancer Research Technology Limited (GB) 2025-09-10 EP claimed
WO-2024094963-A1 2-AMINO-PYRIDO[2,3-D]PYRIMIDIN-7(8H)-ONE AND 7-AMINO-1-PYRIMIDO[4,5-D]PYRIMIDIN-2(1 H)-ONE DERIVATIVES AS EGFR INHIBITORS FOR THE TREATMENT OF CANCER CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2024-05-10 WO claimed
EP-4612148-A1 2-AMINO-PYRIDO[2,3-D]PYRIMIDIN-7(8H)-ONE AND 7-AMINO-1-PYRIMIDO[4,5-D]PYRIMIDIN-2(1 H)-ONE DERIVATIVES AS EGFR INHIBITORS FOR THE TREATMENT OF CANCER Cancer Research Technology Limited (GB) 2025-09-10 EP disclosed
WO-2024094963-A1 2-AMINO-PYRIDO[2,3-D]PYRIMIDIN-7(8H)-ONE AND 7-AMINO-1-PYRIMIDO[4,5-D]PYRIMIDIN-2(1 H)-ONE DERIVATIVES AS EGFR INHIBITORS FOR THE TREATMENT OF CANCER CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2024-05-10 WO disclosed