SCHEMBL30879263

SCHEMBL30879263

CC(C)[Si](C#Cc1c(-c2ccccc2Cl)c(=O)n(C)c2nc(Nc3cccc(CO)c3)ncc12)(C(C)C)C(C)C

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 10/20 0.59
SRC P12931 9/20 0.59
PDGFRB P09619 8/20 0.59
PDGFRA P16234 8/20 0.59
MAPK14 Q16539 8/20 0.59
EGFR P00533 6/20 0.59
FGFR1 P11362 6/20 0.59
KIT P10721 2/20 0.59
WEE1 P30291 8/20 0.53
FGFR2 P21802 2/20 0.46
FGFR4 P22455 2/20 0.46
FGFR3 P22607 2/20 0.46
RIPK2 O43353 2/20 0.45
ACVR1 Q04771 2/20 0.45
NOD2 Q9HC29 1/20 0.45
BMPR1B O00238 1/20 0.44
STK25 O00506 1/20 0.44
GAK O14976 1/20 0.44
EPHB6 O15197 1/20 0.44
JAK2 O60674 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30878932 0.93 ABL1 (0.62) ABL1SRCPDGFRBPDGFRAMAPK14
SCHEMBL30878311 0.89 SRC (0.67) ABL1SRCPDGFRBPDGFRAMAPK14
SCHEMBL30878861 0.89 WEE1 (0.67) ABL1SRCPDGFRBPDGFRAMAPK14
SCHEMBL30879136 0.87 FGFR1 (0.59) ABL1SRCPDGFRBPDGFRAMAPK14
SCHEMBL30878456 0.81 ABL1 (0.70) ABL1SRCPDGFRBPDGFRAMAPK14
SCHEMBL30878459 0.81 ABL1 (0.65) ABL1SRCPDGFRBPDGFRAMAPK14
SCHEMBL30878665 0.81 WEE1 (0.49) ABL1SRCPDGFRBPDGFRAMAPK14
SCHEMBL30879233 0.81 WEE1 (0.52) ABL1SRCPDGFRBPDGFRAMAPK14
SCHEMBL30878805 0.80 EGFR (0.56) SRCEGFRFGFR1WEE1LCK
SCHEMBL30878753 0.80 SRC (0.58) SRCPDGFRBPDGFRAFGFR1WEE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4612148-A1 2-AMINO-PYRIDO[2,3-D]PYRIMIDIN-7(8H)-ONE AND 7-AMINO-1-PYRIMIDO[4,5-D]PYRIMIDIN-2(1 H)-ONE DERIVATIVES AS EGFR INHIBITORS FOR THE TREATMENT OF CANCER Cancer Research Technology Limited (GB) 2025-09-10 EP disclosed
WO-2024094963-A1 2-AMINO-PYRIDO[2,3-D]PYRIMIDIN-7(8H)-ONE AND 7-AMINO-1-PYRIMIDO[4,5-D]PYRIMIDIN-2(1 H)-ONE DERIVATIVES AS EGFR INHIBITORS FOR THE TREATMENT OF CANCER CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2024-05-10 WO disclosed