SCHEMBL30879301

SCHEMBL30879301

CSc1ncc2c(n1)N(C)C(=O)C(c1ccccc1)C2=O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.37
LMNA P02545 2/20 0.37
TP53 P04637 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
MAPK1 P28482 1/20 0.37
HTR2B P41595 1/20 0.37
FGFR4 P22455 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
ALDH1A1 P00352 4/20 0.34
KDM4E B2RXH2 1/20 0.34
NTRK1 P04629 1/20 0.34
RPS6KA5 O75582 1/20 0.34
CCNA2 P20248 1/20 0.34
CDK2 P24941 1/20 0.34
SLC6A2 P23975 5/20 0.33
CACNA2D1 P54289 5/20 0.33
GFER P55789 1/20 0.33
AKT1 P31749 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30879072 0.83 STK4 (0.38) MAPTLMNATP53CYP1A2FGFR4
SCHEMBL30878982 0.82 RPS6KA5 (0.37) MAPTLMNATP53FGFR4MEN1
SCHEMBL30879176 0.80 KDM4C (0.41) MAPTTP53FGFR4MEN1KMT2A
SCHEMBL30879246 0.78 FGFR4 (0.36) MAPTFGFR4MEN1KMT2AKDM4E
SCHEMBL7590747 0.76 MAPT (0.36) MAPTTP53FGFR4MEN1KMT2A
SCHEMBL17070930 0.68 HPGD (0.57) MAPTLMNATP53CYP1A2CYP3A4
SCHEMBL18186302 0.66 MAPK14 (0.40) MAPTLMNAMEN1KMT2AKDM4E
SCHEMBL30879206 0.66 FGFR4 (0.40) MAPTFGFR4MEN1KMT2AALDH1A1
SCHEMBL3532054 0.66 SLC6A2 (0.38) MAPTLMNAFGFR4MEN1KMT2A
SCHEMBL3745747 0.65 MEN1 (0.36) CYP1A2MEN1KMT2AALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4612148-A1 2-AMINO-PYRIDO[2,3-D]PYRIMIDIN-7(8H)-ONE AND 7-AMINO-1-PYRIMIDO[4,5-D]PYRIMIDIN-2(1 H)-ONE DERIVATIVES AS EGFR INHIBITORS FOR THE TREATMENT OF CANCER Cancer Research Technology Limited (GB) 2025-09-10 EP disclosed
WO-2024094963-A1 2-AMINO-PYRIDO[2,3-D]PYRIMIDIN-7(8H)-ONE AND 7-AMINO-1-PYRIMIDO[4,5-D]PYRIMIDIN-2(1 H)-ONE DERIVATIVES AS EGFR INHIBITORS FOR THE TREATMENT OF CANCER CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2024-05-10 WO disclosed