SCHEMBL30879872

SCHEMBL30879872

COc1cccc(C(N)c2ccccn2)c1

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 1/20 0.45
CLK4 Q9HAZ1 1/20 0.45
ROCK1 Q13464 1/20 0.45
TAAR1 Q96RJ0 2/20 0.44
AHR P35869 1/20 0.42
AOC3 Q16853 3/20 0.42
DRD2 P14416 1/20 0.42
SLC6A2 P23975 1/20 0.42
SLC6A4 P31645 1/20 0.42
SLC6A3 Q01959 1/20 0.42
VDR P11473 1/20 0.42
GRM5 P41594 1/20 0.42
GRM4 Q14833 1/20 0.42
P4HB P07237 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
CASR P41180 1/20 0.40
SLC10A1 Q14973 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17842030 1.00 DYRK1A (0.45) DYRK1ACLK4ROCK1TAAR1AHR
Hydrochloric Acid SCHEMBL17842300 0.98 ROCK1 (0.44) DYRK1ACLK4ROCK1TAAR1AHR
SCHEMBL11722266 0.83 AHR (0.54) CLK4ROCK1AHRSLC6A2SLC6A4
SCHEMBL29518433 0.82 DYRK1A (0.45) DYRK1ACLK4AHRAOC3DRD2
SCHEMBL17842130 0.82 DYRK1A (0.45) DYRK1ACLK4AHRAOC3DRD2
SCHEMBL28557150 0.82 SLC6A3 (0.64) DYRK1ACLK4AHRDRD2SLC6A2
SCHEMBL30879852 0.82 AOC3 (0.42) DYRK1ACLK4ROCK1TAAR1AOC3
SCHEMBL30638827 0.82 SLC6A3 (0.64) DYRK1ACLK4AHRDRD2SLC6A2
SCHEMBL17842041 0.81 GRM5 (0.43) DYRK1ASLC6A2SLC6A4SLC6A3GRM5
SCHEMBL29588451 0.81 DYRK1A (0.44) DYRK1ACLK4AHRDRD2SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024092222-A1 MODULATORS OF MAS-RELATED G-PROTEIN RECEPTOR D AND RELATED PRODUCTS AND METHODS ESCIENT PHARMACEUTICALS, INC. (US) 2024-05-02 WO disclosed