SCHEMBL29588451

SCHEMBL29588451

COc1cccc(C(SC(c2cccc(OC)c2)c2ccccn2)c2ccccn2)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 1/20 0.44
CLK4 Q9HAZ1 1/20 0.44
VDR P11473 1/20 0.44
P4HB P07237 1/20 0.43
SLC10A1 Q14973 1/20 0.42
DRD2 P14416 2/20 0.41
SLC6A2 P23975 1/20 0.41
SLC6A4 P31645 1/20 0.41
SLC6A3 Q01959 1/20 0.41
GRM5 P41594 2/20 0.41
GRM4 Q14833 1/20 0.41
PKM P14618 3/20 0.40
MAPT P10636 2/20 0.40
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
GAA P10253 1/20 0.40
CASR P41180 1/20 0.40
NFE2L2 Q16236 1/20 0.39
NPC1 O15118 3/20 0.39
RAB9A P51151 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL17842300 0.82 ROCK1 (0.44) DYRK1ACLK4VDRP4HBSLC10A1
SCHEMBL17842030 0.81 DYRK1A (0.45) DYRK1ACLK4VDRP4HBSLC10A1
SCHEMBL17842130 0.81 DYRK1A (0.45) DYRK1ACLK4VDRP4HBSLC10A1
SCHEMBL28557150 0.81 SLC6A3 (0.64) DYRK1ACLK4VDRP4HBSLC10A1
SCHEMBL30879872 0.81 DYRK1A (0.45) DYRK1ACLK4VDRP4HBSLC10A1
SCHEMBL30638827 0.81 SLC6A3 (0.64) DYRK1ACLK4VDRP4HBSLC10A1
SCHEMBL29518433 0.81 DYRK1A (0.45) DYRK1ACLK4VDRP4HBSLC10A1
SCHEMBL17858535 0.77 DYRK1A (0.42) DYRK1ACLK4VDRP4HBSLC10A1
SCHEMBL7546358 0.74 PBRM1 (0.46) DYRK1ACLK4VDRSLC10A1DRD2
SCHEMBL28662969 0.72 CASR (0.61) CLK4VDRP4HBDRD2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111559976-B Synthetic method of heteroaryl thioether 扬州大学 2022-05-13 CN disclosed