SCHEMBL30898347

SCHEMBL30898347

FC(F)(F)c1ccc(N2CC3(CNC3)C2)nc1

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.46
LMNA P02545 2/20 0.46
ABL1 P00519 1/20 0.46
MAPT P10636 6/20 0.44
SMN1; SMN2 Q16637 4/20 0.44
GAA P10253 1/20 0.44
HPGD P15428 1/20 0.43
KMT2A Q03164 2/20 0.43
ALDH1A1 P00352 2/20 0.42
CYP3A4 P08684 1/20 0.42
MEN1 O00255 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
EIF2AK4 Q9P2K8 1/20 0.42
L3MBTL1 Q9Y468 3/20 0.42
APAF1 O14727 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
HTT P42858 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25145868 1.00 KDM4E (0.46) KDM4ELMNAABL1MAPTSMN1; SMN2
SCHEMBL31239676 0.80 HSD17B10 (0.40) SMN1; SMN2HPGDALDH1A1CYP3A4CYP1A2
SCHEMBL20798102 0.80 AVPR1A (0.44) HPGDALDH1A1CYP3A4CYP1A2
SCHEMBL485461 0.79 KCNH2 (0.48) KDM4ELMNAABL1MAPTSMN1; SMN2
Hydrochloric Acid SCHEMBL25309482 0.78 HSD17B10 (0.39) SMN1; SMN2HPGDALDH1A1CYP3A4CYP1A2
SCHEMBL25145697 0.77 PARP1 (0.38) HPGDALDH1A1CYP1A2EIF2AK4
SCHEMBL231823 0.76 ADRB1 (0.60) KDM4ELMNAABL1MAPTSMN1; SMN2
SCHEMBL20511824 0.76 GRIN2D (0.44) HPGDALDH1A1CYP3A4CYP1A2CYP2C9
SCHEMBL17035908 0.76 ADRB1 (0.60) KDM4ELMNAABL1MAPTSMN1; SMN2
SCHEMBL31541438 0.76 GRIN2D (0.44) HPGDALDH1A1CYP3A4CYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118103374-A Heterocyclic compounds 豪夫迈·罗氏有限公司 2024-05-28 CN disclosed