SCHEMBL30900367

SCHEMBL30900367

FC(F)(F)Oc1ccc(I)cc1Br

nearest known ligand 0.34

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.34
ALDH1A1 P00352 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
EPHX2 P34913 2/20 0.34
MBOAT4 Q96T53 1/20 0.34
PDE2A O00408 1/20 0.32
TRPV1 Q8NER1 1/20 0.32
SLC1A5 Q15758 2/20 0.31
PNMT P11086 3/20 0.31
MGLL Q99685 1/20 0.31
TSHR P16473 1/20 0.31
ALOX15 P16050 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21648919 1.00 MAPK1 (0.34) MAPK1ALDH1A1TDP1L3MBTL1EPHX2
SCHEMBL20309114 0.84 TRPV1 (0.32) EPHX2TRPV1SLC1A5PNMT
SCHEMBL19033849 0.78 EPHX2 (0.50) EPHX2PDE2ATRPV1SLC1A5
SCHEMBL261397 0.78 PKM (0.47) MAPK1ALDH1A1TDP1L3MBTL1EPHX2
SCHEMBL24731505 0.76 MAPK1 (0.34) MAPK1ALDH1A1TDP1L3MBTL1EPHX2
SCHEMBL17420405 0.76 SCN5A (0.41) EPHX2PDE2ATRPV1SLC1A5
SCHEMBL508527 0.76 SLC1A5 (0.47) SLC1A5
SCHEMBL16951248 0.76 MBOAT4 (0.36) MAPK1ALDH1A1TDP1L3MBTL1EPHX2
SCHEMBL263399 0.76 EPHX2 (0.38) MAPK1ALDH1A1TDP1L3MBTL1EPHX2
SCHEMBL263489 0.76 MBOAT4 (0.39) MAPK1ALDH1A1TDP1L3MBTL1EPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117658987-A Compounds as PLK1 inhibitors, and preparation method and application thereof 上海深势唯思科技有限责任公司 2024-03-08 CN disclosed