SCHEMBL30902253

SCHEMBL30902253

COc1ncc(Br)cc1NS(=O)(=O)c1ccc(F)cc1Cl

nearest known ligand 0.55

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 19/20 0.55
PIK3CD O00329 2/20 0.52
PIK3CB P42338 2/20 0.52
PIK3R1 P27986 2/20 0.52
MTOR P42345 2/20 0.52
PIK3CG P48736 1/20 0.52
CCR4 P51679 1/20 0.50
CYP3A4 P08684 1/20 0.49
CYP2C9 P11712 1/20 0.49
CYP2C19 P33261 1/20 0.49
KCNH2 Q12809 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30333881 0.88 PIK3CA (0.59) PIK3CAPIK3CDPIK3CBPIK3R1MTOR
SCHEMBL462714 0.88 PIK3CA (0.59) PIK3CAPIK3CDPIK3CBPIK3R1MTOR
SCHEMBL29610307 0.88 PIK3CA (0.59) PIK3CAPIK3CDPIK3CBPIK3R1MTOR
SCHEMBL22447740 0.88 ACLY (0.46) PIK3CAPIK3CDPIK3CBPIK3R1MTOR
SCHEMBL22447679 0.87 PIK3CA (0.49) PIK3CAPIK3CDPIK3CBPIK3R1MTOR
SCHEMBL22447379 0.85 MEN1 (0.50) PIK3CA
SCHEMBL2919328 0.84 PIK3CD (0.54) PIK3CAPIK3CDPIK3CBMTORPIK3CG
SCHEMBL15556197 0.82 MTOR (0.55) PIK3CAPIK3CDPIK3CBPIK3R1MTOR
SCHEMBL22447736 0.81 CCR4 (0.64) CCR4
SCHEMBL22447698 0.81 PIK3CA (0.53) PIK3CAPIK3CDPIK3CBPIK3R1MTOR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117957219-A Pyridine derivative and application thereof 四川汇宇制药股份有限公司 2024-04-30 CN disclosed