SCHEMBL30929470

SCHEMBL30929470

Cc1cc(C)cc(CNc2cnc3n(c2=O)[C@H](C(=O)NCc2cccnc2C)CC3)c1

nearest known ligand 0.51

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
F2 P00734 2/20 0.51
F7 P08709 1/20 0.51
F3 P13726 1/20 0.51
P2RX7 Q99572 15/20 0.41
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
GAA P10253 1/20 0.40
PIK3CA P42336 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30929396 0.87 F2 (0.51) F2F7F3
SCHEMBL30929412 0.84 F2 (0.54) F2F7F3P2RX7CYP3A4
SCHEMBL30929436 0.82 F2 (0.57) F2F7F3P2RX7CYP3A4
SCHEMBL30929392 0.81 F2 (0.49) F2F7F3
SCHEMBL30929426 0.81 F2 (0.52) F2F7F3P2RX7CYP3A4
SCHEMBL30929472 0.81 F2 (0.44) F2F7F3P2RX7CYP3A4
SCHEMBL30929399 0.81 F2 (0.47) F2F7F3P2RX7CYP3A4
SCHEMBL30929425 0.81 F2 (0.47) F2F7F3
SCHEMBL30929397 0.80 F2 (0.47) F2F7F3P2RX7
SCHEMBL30929415 0.77 F2 (0.44) F2F7F3CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4626891-A1 FUSED PYRIMIDINES AS MASP-2 INHIBITORS Omeros Corporation (US) 2025-10-08 EP disclosed
WO-2024118840-A1 FUSED PYRIMIDINES AS MASP-2 INHIBITORS OMEROS CORPORATION (US) 2024-06-06 WO disclosed