SCHEMBL30929426

SCHEMBL30929426

Cc1cc(C)cc(CNc2cnc3n(c2=O)[C@H](C(=O)NCc2cncc(Cl)c2)CC3)c1

nearest known ligand 0.52

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
F2 P00734 4/20 0.52
F7 P08709 4/20 0.52
F3 P13726 4/20 0.52
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
P2RX7 Q99572 6/20 0.38
KMT2A Q03164 1/20 0.37
CFD P00746 2/20 0.36
PREP P48147 3/20 0.36
WDR5 P61964 1/20 0.35
F10 P00742 2/20 0.35
SSTR2 P30874 1/20 0.34
KCNH2 Q12809 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30929412 0.84 F2 (0.54) F2F7F3CYP3A4CYP2C9
SCHEMBL30929436 0.83 F2 (0.57) F2F7F3CYP3A4CYP2C9
SCHEMBL30929414 0.83 F2 (0.48) F2F7F3CYP3A4CYP2C9
SCHEMBL30929405 0.83 F2 (0.46) F2F7F3CYP3A4CYP2C9
SCHEMBL30929477 0.82 F2 (0.49) F2F7F3CYP3A4CYP2C9
SCHEMBL30929452 0.82 F2 (0.45) F2F7F3P2RX7KMT2A
SCHEMBL30929399 0.82 F2 (0.47) F2F7F3CYP3A4CYP2C9
SCHEMBL30929422 0.82 F2 (0.52) F2F7F3CYP3A4CYP2C9
SCHEMBL30929470 0.81 F2 (0.51) F2F7F3CYP3A4CYP2C9
SCHEMBL30929395 0.81 F2 (0.47) F2F7F3CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4626891-A1 FUSED PYRIMIDINES AS MASP-2 INHIBITORS Omeros Corporation (US) 2025-10-08 EP disclosed
WO-2024118840-A1 FUSED PYRIMIDINES AS MASP-2 INHIBITORS OMEROS CORPORATION (US) 2024-06-06 WO disclosed