SCHEMBL3093252

SCHEMBL3093252

Cc1c(C(=O)NN2CCCCC2)nc(-c2ccc(Cl)cc2Cl)n1-c1ccc(OS(=O)(=O)CCCC(F)(F)F)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 20/20 1.00
CNR2 P34972 4/20 0.69

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4243002 0.99 CNR1 (0.99) CNR1CNR2
Sulfuric Acid SCHEMBL4242588 0.99 CNR1 (0.97) CNR1CNR2
SCHEMBL4242278 0.97 CNR1 (0.93) CNR1CNR2
SCHEMBL3093160 0.96 CNR1 (1.00) CNR1CNR2
SCHEMBL29473535 0.96 CNR1 (1.00) CNR1CNR2
Hydrochloric Acid SCHEMBL4248848 0.95 CNR1 (0.98) CNR1CNR2
SCHEMBL4245868 0.94 CNR1 (0.97) CNR1CNR2
Sulfuric Acid SCHEMBL4241613 0.94 CNR1 (0.97) CNR1CNR2
SCHEMBL4246768 0.93 CNR1 (0.94) CNR1CNR2
SCHEMBL4616800 0.92 CNR1 (1.00) CNR1CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7799804-B2 Therapeutic agents ASTRAZENECA AB (SE) 2010-09-21 US claimed
US-20090005415-A1 1,2-Diarylimidazoles for Use as Cb1 Modulators ASTRAZENECA AB (SE) 2009-01-01 US claimed
EP-1940803-A1 1,2-DIARYLIMIDAZOLES FOR USE AS CBI MODULATORS AstraZeneca AB (SE) 2008-07-09 EP claimed
US-20070208059-A1 Therapeutic Agents ASTRAZENECA AB (SE) 2007-09-06 US claimed
WO-2007031720-A1 1,2-DIARYLIMIDAZOLES FOR USE AS CBI MODULATORS ASTRAZENECA AB (SE) 2007-03-22 WO claimed
US-7799804-B2 Therapeutic agents ASTRAZENECA AB (SE) 2010-09-21 US disclosed
US-20090005415-A1 1,2-Diarylimidazoles for Use as Cb1 Modulators ASTRAZENECA AB (SE) 2009-01-01 US disclosed
EP-1940803-A1 1,2-DIARYLIMIDAZOLES FOR USE AS CBI MODULATORS AstraZeneca AB (SE) 2008-07-09 EP disclosed
US-20070208059-A1 Therapeutic Agents ASTRAZENECA AB (SE) 2007-09-06 US disclosed
WO-2007031720-A1 1,2-DIARYLIMIDAZOLES FOR USE AS CBI MODULATORS ASTRAZENECA AB (SE) 2007-03-22 WO disclosed
EP-1735287-A1 THERAPEUTIC AGENTS Astrazeneca AB (SE) 2006-12-27 EP disclosed
WO-2005095354-A1 THERAPEUTIC AGENTS ASTRAZENECA AB (SE) 2005-10-13 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090005415-A1 1,2-Diarylimidazoles for Use as Cb1 Modulators CNR2, CNR1, FAAH CNR1 2/4885CNR2 1/4885
US-20070208059-A1 Therapeutic Agents NLN, BDNF, GAP43 CNR1 193/4885CNR2 254/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.