SCHEMBL30935191

SCHEMBL30935191

C=CC(=O)Nc1cccc(B(O)O)c1

nearest known ligand 0.61

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TGM2 P21980 7/20 0.61
TRPV1 Q8NER1 1/20 0.58
BTK Q06187 3/20 0.58
JAK3 P52333 3/20 0.48
JAK2 O60674 1/20 0.48
NLRP3 Q96P20 1/20 0.48
F13A1 P00488 1/20 0.46
LMNA P02545 1/20 0.46
TGM1 P22735 1/20 0.46
TGM3 Q08188 1/20 0.46
EGFR P00533 1/20 0.46
MAP2K7 O14733 1/20 0.46
AURKA O14965 1/20 0.46
ESRRG P62508 2/20 0.45
ESR1 P03372 1/20 0.45
ESR2 Q92731 1/20 0.45
LPAR1 Q92633 1/20 0.45
LPAR2 Q9HBW0 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL235432 1.00 TGM2 (0.61) TGM2TRPV1BTKJAK3JAK2
SCHEMBL29246639 0.98 TGM2 (0.59) TGM2TRPV1BTKJAK3JAK2
Acrylamide SCHEMBL22206248 0.94 TGM2 (0.55) TGM2TRPV1BTKJAK3JAK2
Acrylamide SCHEMBL30480310 0.94 TGM2 (0.55) TGM2TRPV1BTKJAK3JAK2
SCHEMBL23199033 0.89 TDP1 (0.54) TGM2TRPV1BTKJAK3JAK2
SCHEMBL30480308 0.89 TGM2 (0.50) TGM2TRPV1BTKJAK3JAK2
SCHEMBL18100115 0.87 TGM2 (0.58) TGM2TRPV1BTKJAK3F13A1
SCHEMBL4103284 0.84 TGM2 (0.76) TGM2BTKJAK3F13A1LMNA
SCHEMBL16193308 0.83 TGM2 (0.54) TGM2TRPV1BTKJAK3F13A1
SCHEMBL11349846 0.81 TRPV1 (0.51) TRPV1BTKNLRP3ESRRGESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024125464-A1 TETRAHYDROISOQUINOLIN-ONE DERIVATIVES, PREPARATION METHODS AND MEDICINAL USES THEREOF JIANGSU HANSOH PHARMACEUTICAL GROUP CO., LTD. (CN) 2024-06-20 WO disclosed