SCHEMBL30940499

SCHEMBL30940499

[2H]C([2H])([2H])NC(=O)c1nncc(Nc2ccc(C(F)F)nn2)c1Nc1ncccc1S(C)(=O)=O

nearest known ligand 0.44

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TYK2 P29597 20/20 0.44
JAK1 P23458 6/20 0.44
JAK2 O60674 4/20 0.44
JAK3 P52333 1/20 0.44
STAT3 P40763 1/20 0.39
KCNH2 Q12809 3/20 0.34
UGT1A1 P22309 1/20 0.32
KIT P10721 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30940481 0.89 TYK2 (0.46) TYK2JAK1JAK2JAK3STAT3
SCHEMBL20985299 0.84 TYK2 (0.61) TYK2JAK1JAK2JAK3STAT3
SCHEMBL30940516 0.79 TYK2 (0.42) TYK2JAK1JAK2JAK3STAT3
SCHEMBL30617391 0.76 TYK2 (0.62) TYK2JAK1JAK2JAK3STAT3
SCHEMBL20985233 0.76 TYK2 (0.62) TYK2JAK1JAK2JAK3STAT3
SCHEMBL30940500 0.75 TYK2 (0.36) TYK2JAK1JAK2JAK3KCNH2
SCHEMBL30617361 0.75 TYK2 (0.40) TYK2JAK1JAK2JAK3STAT3
SCHEMBL30940517 0.74 TYK2 (0.53) TYK2JAK1JAK2JAK3STAT3
SCHEMBL20985231 0.74 TYK2 (0.63) TYK2JAK1JAK2JAK3STAT3
SCHEMBL30940487 0.74 TYK2 (0.39) TYK2JAK1JAK2JAK3KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111315737-B Heteroaryl compounds substituted with sulfone pyridinylalkylamides 百时美施贵宝公司 2024-06-18 CN disclosed