SCHEMBL30940487

SCHEMBL30940487

COc1ccc(Nc2cnnc(C(N)=O)c2Nc2ncccc2S(C)(=O)=O)nn1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TYK2 P29597 11/20 0.39
JAK1 P23458 6/20 0.39
CA12 O43570 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA9 Q16790 1/20 0.35
JAK2 O60674 5/20 0.34
JAK3 P52333 3/20 0.34
LMNA P02545 2/20 0.33
LRRK2 Q5S007 1/20 0.33
KCNH2 Q12809 2/20 0.33
SYK P43405 1/20 0.33
KIT P10721 1/20 0.33
NNMT P40261 1/20 0.32
EDNRA P25101 1/20 0.32
SMN1; SMN2 Q16637 2/20 0.31
NPC1 O15118 1/20 0.31
MAPT P10636 1/20 0.31
AHR P35869 1/20 0.31
RAB9A P51151 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20985227 0.82 TYK2 (0.48) TYK2JAK1CA12CA1CA2
SCHEMBL30940512 0.79 TYK2 (0.41) TYK2JAK1LMNASMN1; SMN2NPC1
SCHEMBL30940530 0.77 TYK2 (0.39) TYK2JAK1JAK2JAK3LMNA
SCHEMBL30940499 0.74 TYK2 (0.44) TYK2JAK1JAK2JAK3KCNH2
SCHEMBL20985238 0.74 TYK2 (0.61) TYK2JAK1JAK2JAK3KCNH2
SCHEMBL30940531 0.74 TYK2 (0.61) TYK2JAK1JAK2JAK3KCNH2
SCHEMBL30940528 0.74 TYK2 (0.45) TYK2JAK1JAK2JAK3LMNA
SCHEMBL30940481 0.72 TYK2 (0.46) TYK2JAK1JAK2JAK3KCNH2
SCHEMBL30617400 0.72 TYK2 (0.63) TYK2JAK1JAK2JAK3KCNH2
SCHEMBL24587279 0.71 TYK2 (0.48) TYK2JAK1JAK2JAK3SYK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111315737-B Heteroaryl compounds substituted with sulfone pyridinylalkylamides 百时美施贵宝公司 2024-06-18 CN disclosed