SCHEMBL30944359

SCHEMBL30944359

CC12CC3CC(C)(C1)CC(C(=O)Nc1nc4cc(C(F)(F)F)ccc4s1)(C3)C2

nearest known ligand 0.58

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 2/20 0.58
NCS1 P62166 1/20 0.48
CNR1 P21554 1/20 0.48
CYP2D6 P10635 1/20 0.46
NPC1 O15118 3/20 0.44
RAB9A P51151 3/20 0.44
CSNK1D P48730 5/20 0.44
ADORA1 P30542 1/20 0.44
ALOX15 P16050 1/20 0.43
GAA P10253 1/20 0.43
HTT P42858 1/20 0.43
ACP1 P24666 1/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
RXFP1 Q9HBX9 1/20 0.41
CLK1 P49759 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28520781 1.00 DYRK1A (0.58) DYRK1ANCS1CNR1CYP2D6NPC1
SCHEMBL28530647 0.92 DYRK1A (0.58) DYRK1ACNR1CYP2D6NPC1RAB9A
SCHEMBL30944301 0.92 DYRK1A (0.58) DYRK1ACNR1CYP2D6NPC1RAB9A
SCHEMBL30944318 0.92 DYRK1A (0.58) DYRK1ACNR1CYP2D6NPC1RAB9A
SCHEMBL30944406 0.87 DYRK1A (0.56) DYRK1ACNR1NPC1RAB9ACSNK1D
SCHEMBL30944415 0.85 ADORA1 (0.62) DYRK1ACNR1CYP2D6NPC1RAB9A
SCHEMBL30944351 0.85 CNR1 (0.51) DYRK1ACNR1CYP2D6NPC1RAB9A
SCHEMBL30944407 0.83 NPC1 (0.50) CNR1NPC1RAB9ACSNK1DADORA1
SCHEMBL30944393 0.82 CNR1 (0.71) DYRK1ACNR1NPC1RAB9ACSNK1D
SCHEMBL31236381 0.81 NPC1 (0.66) DYRK1ACNR1NPC1RAB9AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118772080-A Antimycobacterial heterocyclic amides 克莱斯通公司 2024-10-15 CN claimed
CN-118772080-A Antimycobacterial heterocyclic amides 克莱斯通公司 2024-10-15 CN disclosed
CN-112423746-B Novel antimycobacterial heterocyclic amides 克莱斯通公司 2024-06-28 CN disclosed