SCHEMBL30944407

SCHEMBL30944407

CC12CC3CC(C)(C1)CC(C(=O)Nc1nc4cc(F)c(F)cc4s1)(C3)C2

nearest known ligand 0.55

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.50
RAB9A P51151 3/20 0.50
CNR1 P21554 1/20 0.47
ALOX15 P16050 1/20 0.47
GAA P10253 1/20 0.47
HTT P42858 1/20 0.47
CLK1 P49759 1/20 0.44
P2RX7 Q99572 1/20 0.41
ADORA1 P30542 2/20 0.41
ADORA2A P29274 1/20 0.41
CSNK1D P48730 1/20 0.40
CSNK1E P49674 1/20 0.40
KMT2A Q03164 2/20 0.40
MEN1 O00255 1/20 0.40
RXFP1 Q9HBX9 1/20 0.40
LMNA P02545 1/20 0.39
MAPT P10636 1/20 0.39
POLB P06746 1/20 0.39
TRPV1 Q8NER1 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31236381 0.87 NPC1 (0.66) NPC1RAB9ACNR1GAAHTT
SCHEMBL30944406 0.87 DYRK1A (0.56) NPC1RAB9ACNR1ALOX15GAA
SCHEMBL28530631 0.84 DYRK1A (0.55) NPC1RAB9ACNR1HTTCLK1
SCHEMBL30944384 0.84 DYRK1A (0.55) NPC1RAB9ACNR1HTTCLK1
SCHEMBL30944410 0.84 GAA (0.47) NPC1RAB9ACNR1ALOX15GAA
SCHEMBL30944383 0.83 DYRK1A (0.56) NPC1RAB9ACNR1CLK1KMT2A
SCHEMBL30944415 0.83 ADORA1 (0.62) NPC1RAB9ACNR1ALOX15GAA
SCHEMBL30944300 0.83 RAB9A (0.56) NPC1RAB9ACNR1ALOX15GAA
SCHEMBL30944419 0.83 RAB9A (0.56) NPC1RAB9ACNR1GAAHTT
SCHEMBL30944351 0.83 CNR1 (0.51) NPC1RAB9ACNR1ALOX15GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118772080-A Antimycobacterial heterocyclic amides 克莱斯通公司 2024-10-15 CN claimed
CN-118772080-A Antimycobacterial heterocyclic amides 克莱斯通公司 2024-10-15 CN disclosed
CN-112423746-B Novel antimycobacterial heterocyclic amides 克莱斯通公司 2024-06-28 CN disclosed