SCHEMBL30948583

SCHEMBL30948583

CN(C)C1CCC2(CC1)CCN(c1ccc(Nc3ncc(Cl)c(Nc4ccccc4P(C)C)n3)cc1N)CC2

nearest known ligand 0.53

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
EGFR P00533 11/20 0.53
ALK Q9UM73 7/20 0.51
AXL P30530 1/20 0.46
MAPK9 P45984 3/20 0.44
MAPK10 P53779 3/20 0.44
CTSC P53634 1/20 0.43
MAPK8 P45983 1/20 0.42
AURKA O14965 1/20 0.42
INSR P06213 1/20 0.42
IGF1R P08069 1/20 0.42
ROS1 P08922 1/20 0.42
EML4 Q9HC35 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30948584 1.00 EGFR (0.53) EGFRALKAXLMAPK9MAPK10
SCHEMBL30948623 0.93 EGFR (0.50) EGFRALKAXLMAPK9MAPK10
SCHEMBL30948582 0.93 EGFR (0.50) EGFRALKAXLMAPK9MAPK10
SCHEMBL30948615 0.88 ALK (0.55) EGFRALKAURKAINSRIGF1R
SCHEMBL22246247 0.87 EGFR (0.52) EGFRALKAXLMAPK9MAPK10
SCHEMBL30948600 0.87 EGFR (0.49) EGFRALKMAPK9MAPK10MAPK8
SCHEMBL22520091 0.87 EGFR (0.60) EGFRALKAURKAINSRIGF1R
SCHEMBL22246279 0.85 EGFR (0.60) EGFRALKAXLMAPK9MAPK10
SCHEMBL22246241 0.84 EGFR (0.49) EGFRALKAXLMAPK9MAPK10
SCHEMBL30948622 0.83 EGFR (0.59) EGFRALKAXL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113677680-B EGFR inhibitor, composition and application thereof 贝达药业股份有限公司 2024-05-10 CN disclosed