SCHEMBL30948600

SCHEMBL30948600

CN1CC2(CCN(c3ccc(Nc4ncc(Cl)c(Nc5ccccc5P(C)C)n4)cc3N)CC2)C1

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
EGFR P00533 7/20 0.49
CCNK O75909 2/20 0.47
CCNA2 P20248 2/20 0.47
CDK2 P24941 2/20 0.47
CCND3 P30281 2/20 0.47
CDK9 P50750 2/20 0.47
CDK6 Q00534 2/20 0.47
MAPK9 P45984 3/20 0.46
MAPK10 P53779 3/20 0.46
SLC2A1 P11166 2/20 0.46
ALK Q9UM73 6/20 0.46
MAPK8 P45983 1/20 0.45
MAP3K7 O43318 1/20 0.44
FGFR1 P11362 1/20 0.44
SRC P12931 1/20 0.44
MAPK1 P28482 1/20 0.44
MAP2K1 Q02750 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22246172 0.91 MAPK9 (0.54) EGFRCCNKCCNA2CDK2CCND3
SCHEMBL30948622 0.90 EGFR (0.59) EGFRCCNKCCNA2CDK2CCND3
SCHEMBL30948623 0.88 EGFR (0.50) EGFRCCNKCCNA2CDK2CCND3
SCHEMBL30948584 0.87 EGFR (0.53) EGFRMAPK9MAPK10ALKMAPK8
SCHEMBL30948583 0.87 EGFR (0.53) EGFRMAPK9MAPK10ALKMAPK8
SCHEMBL22520147 0.86 EGFR (0.68) EGFRALK
SCHEMBL30948582 0.85 EGFR (0.50) EGFRCCNA2CDK2MAPK9MAPK10
SCHEMBL22246276 0.84 EGFR (0.49) EGFRCCNKCCNA2CDK2CCND3
SCHEMBL22246232 0.82 MAPK9 (0.55) EGFRCCNKCCNA2CDK2CCND3
SCHEMBL30503703 0.82 MAPK9 (0.55) EGFRCCNKCCNA2CDK2CCND3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113677680-B EGFR inhibitor, composition and application thereof 贝达药业股份有限公司 2024-05-10 CN disclosed