SCHEMBL30948620

SCHEMBL30948620

CP(C)c1ccccc1Nc1nc(Nc2ccc(N3CCN4CCC[C@H]4C3)c([N+](=O)[O-])c2)ncc1Cl

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
EGFR P00533 12/20 0.49
BRD4 O60885 1/20 0.45
CTSC P53634 1/20 0.44
INSR P06213 1/20 0.44
IGF1R P08069 1/20 0.44
ALK Q9UM73 1/20 0.44
CCNA2 P20248 3/20 0.43
CDK2 P24941 3/20 0.43
CCNK O75909 2/20 0.42
CCND3 P30281 2/20 0.42
CDK9 P50750 2/20 0.42
CDK6 Q00534 2/20 0.42
MAP3K7 O43318 1/20 0.42
FGFR1 P11362 1/20 0.42
SRC P12931 1/20 0.42
MAPK1 P28482 1/20 0.42
MAP2K1 Q02750 1/20 0.42
MAPK9 P45984 1/20 0.41
MAPK10 P53779 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28662985 0.88 EGFR (0.65) EGFRINSRIGF1RALKFGFR1
SCHEMBL28662982 0.88 EGFR (0.65) EGFRINSRIGF1RALKFGFR1
SCHEMBL30948591 0.81 MAPK9 (0.44) EGFRBRD4ALKMAPK9MAPK10
SCHEMBL28665507 0.78 MAPK9 (0.46) BRD4ALKCCNA2CDK2CCNK
SCHEMBL29190558 0.78 ULK1 (0.45) BRD4ALKCCNA2CDK2CCNK
SCHEMBL28667751 0.76 EGFR (0.68) EGFRINSRIGF1RALKFGFR1
SCHEMBL29783086 0.76 EGFR (0.68) EGFRINSRIGF1RALKFGFR1
SCHEMBL30948585 0.76 CCNK (0.52) EGFRBRD4ALKCCNA2CDK2
SCHEMBL28648152 0.76 EGFR (0.84) EGFRINSRIGF1RALKFGFR1
SCHEMBL22520094 0.74 EGFR (0.65) EGFRINSRIGF1RALK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113677680-B EGFR inhibitor, composition and application thereof 贝达药业股份有限公司 2024-05-10 CN disclosed