SCHEMBL30948591

SCHEMBL30948591

CP(C)c1ccccc1Nc1nc(Nc2ccc(N3CCC4(CC3)CC(N)C4)c([N+](=O)[O-])c2)ncc1Cl

nearest known ligand 0.44

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MAPK9 P45984 3/20 0.44
MAPK10 P53779 3/20 0.44
EGFR P00533 9/20 0.44
MAPK8 P45983 1/20 0.43
ALK Q9UM73 7/20 0.42
BRD4 O60885 1/20 0.42
SLC2A1 P11166 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22246276 0.90 EGFR (0.49) MAPK9MAPK10EGFRMAPK8ALK
SCHEMBL22246232 0.88 MAPK9 (0.55) MAPK9MAPK10EGFRMAPK8ALK
SCHEMBL30503703 0.88 MAPK9 (0.55) MAPK9MAPK10EGFRMAPK8ALK
SCHEMBL22246265 0.85 EGFR (0.53) MAPK9MAPK10EGFRMAPK8ALK
SCHEMBL30948585 0.85 CCNK (0.52) MAPK9MAPK10EGFRMAPK8ALK
Trifluoroacetic Acid SCHEMBL29065781 0.84 MAPK9 (0.55) MAPK9MAPK10EGFRMAPK8ALK
SCHEMBL30503700 0.83 EGFR (0.48) MAPK9MAPK10EGFRMAPK8ALK
SCHEMBL22246247 0.81 EGFR (0.52) MAPK9MAPK10EGFRMAPK8ALK
SCHEMBL22520178 0.81 ALK (0.44) EGFRALK
SCHEMBL30948620 0.81 EGFR (0.49) MAPK9MAPK10EGFRALKBRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113677680-B EGFR inhibitor, composition and application thereof 贝达药业股份有限公司 2024-05-10 CN disclosed