SCHEMBL30953732

SCHEMBL30953732

Nc1nc2c(s1)Cc1cc(C(F)(F)F)ccc1-2

nearest known ligand 0.58

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 17/20 0.58
CHEK1 O14757 1/20 0.57
DAPK3 O43293 1/20 0.57
LTK P29376 1/20 0.57
MAPK8 P45983 1/20 0.57
CSNK1A1 P48729 1/20 0.57
CDK8 P49336 1/20 0.57
LIMK1 P53667 1/20 0.57
CDK5 Q00535 1/20 0.57
DYRK1A Q13627 1/20 0.57
LRRK2 Q5S007 1/20 0.57
CLK4 Q9HAZ1 1/20 0.57
DYRK1B Q9Y463 1/20 0.57
FBP1 P09467 2/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30953877 0.89 ADORA1 (0.60) ADORA1CHEK1DAPK3LTKMAPK8
SCHEMBL5573260 0.78 ADORA1 (0.67) ADORA1CHEK1DAPK3LTKMAPK8
SCHEMBL30953825 0.77 KDM4E (0.60) ADORA1CHEK1DAPK3LTKMAPK8
Iodide SCHEMBL4960121 0.77 ADORA1 (0.69) ADORA1CHEK1DAPK3LTKMAPK8
Iodide SCHEMBL3989408 0.77 ADORA1 (0.64) ADORA1CHEK1DAPK3LTKMAPK8
SCHEMBL30953799 0.75 FBP1 (0.46) ADORA1FBP1
SCHEMBL4959991 0.73 CHEK1 (1.00) ADORA1CHEK1DAPK3LTKMAPK8
SCHEMBL31321386 0.73 CHEK1 (1.00) ADORA1CHEK1DAPK3LTKMAPK8
Iodide SCHEMBL3994593 0.73 ADORA1 (1.00) ADORA1CHEK1DAPK3LTKMAPK8
Iodide SCHEMBL3990143 0.73 ADORA1 (0.78) ADORA1CHEK1DAPK3LTKMAPK8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024140431-A1 COMPOUNDS COMPRISING HETEROARYL RINGS AND COMPOSITIONS AND METHODS THEREOF IONGEN THERAPEUTICS CO., LTD. (CN) 2024-07-04 WO disclosed