SCHEMBL30955650

SCHEMBL30955650

CC(C)N1C(=O)N(c2cnc(N)c(F)c2)Cc2cnc(NC3CCC(N(C)C)CC3)nc21

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 2/20 0.38
TNK2 Q07912 2/20 0.36
MAP4K2 Q12851 2/20 0.36
FGFR4 P22455 7/20 0.35
MAPK8 P45983 2/20 0.34
MAPK10 P53779 2/20 0.34
IRAK4 Q9NWZ3 2/20 0.32
FGFR1 P11362 2/20 0.32
FGFR2 P21802 2/20 0.32
FGFR3 P22607 2/20 0.32
CDK4 P11802 3/20 0.32
CCND1 P24385 3/20 0.32
CDK2 P24941 3/20 0.32
CCNT1 O60563 1/20 0.32
CCNA2 P20248 1/20 0.32
CCND3 P30281 1/20 0.32
CDK9 P50750 1/20 0.32
CDK6 Q00534 1/20 0.32
MAPK9 P45984 1/20 0.32
MAPK1 P28482 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30955652 0.89 ERN1 (0.39) ERN1TNK2MAP4K2FGFR4MAPK8
SCHEMBL30955648 0.85 MAPK8 (0.37) ERN1TNK2MAP4K2FGFR4MAPK8
SCHEMBL30955617 0.82 ERN1 (0.41) ERN1TNK2MAP4K2FGFR4MAPK1
SCHEMBL30955556 0.82 ERN1 (0.43) ERN1TNK2MAP4K2FGFR4MAPK8
SCHEMBL30955563 0.82 ERN1 (0.54) ERN1TNK2MAP4K2FGFR4MAPK8
SCHEMBL30955598 0.82 ERN1 (0.47) ERN1TNK2MAP4K2FGFR4CDK2
SCHEMBL30955548 0.81 ERN1 (0.43) ERN1TNK2MAP4K2FGFR4MAPK8
SCHEMBL30955561 0.81 ERN1 (0.43) ERN1TNK2MAP4K2FGFR4MAPK8
SCHEMBL30955501 0.81 ERN1 (0.39) ERN1TNK2MAP4K2FGFR4MAPK8
SCHEMBL30955499 0.78 TNK2 (0.47) TNK2MAP4K2FGFR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024131893-A1 IRE1α SMALL MOLECULE INHIBITORS SHANGHAI YI ZHONG XING BIOTECHNOLOGY CO., LTD. (CN) 2024-06-27 WO disclosed