SCHEMBL30959345

SCHEMBL30959345

CC(C)[Si](C#Cc1cccc2[nH]ncc12)(C(C)C)C(C)C

nearest known ligand 0.55

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.45
NOS1 P29475 4/20 0.44
AXL P30530 2/20 0.44
METAP2 P50579 2/20 0.41
MET P08581 1/20 0.40
JAK2 O60674 1/20 0.39
JAK1 P23458 1/20 0.39
HAO1 Q9UJM8 2/20 0.39
BRD4 O60885 1/20 0.36
TRPV1 Q8NER1 4/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4055516 0.83 IDO1 (0.53) IDO1NOS1AXLMETAP2MET
SCHEMBL30135663 0.79 IDO1 (0.51) IDO1NOS1AXLMETAP2MET
SCHEMBL26259570 0.78 CACNA2D1 (0.36)
SCHEMBL12405326 0.77 CACNA2D1 (0.35)
SCHEMBL30135671 0.75 IDO1 (0.47) IDO1NOS1AXLMETAP2MET
SCHEMBL25238925 0.75 ALK (0.40) JAK2BRD4
SCHEMBL31140667 0.75 ALK (0.40) JAK2BRD4
SCHEMBL29977301 0.72 GRM5 (0.45)
SCHEMBL26259230 0.72 GRM5 (0.45)
SCHEMBL12525231 0.72 NOS1 (0.46) IDO1NOS1AXLMETAP2MET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4615847-A1 SMALL MOLECULE INHIBITORS OF KRAS PROTEINS Merck Sharp & Dohme LLC (US) 2025-09-17 EP disclosed
WO-2024103010-A1 SMALL MOLECULE INHIBITORS OF KRAS PROTEINS MERCK SHARP & DOHME LLC (US) 2024-05-16 WO disclosed