SCHEMBL30964273

SCHEMBL30964273

O=C1Cc2ccc(OCCCCN3CCN(c4cccc(C(F)(F)F)c4)CC3)cc2N1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 14/20 0.66
HTR2A P28223 2/20 0.55
DRD3 P35462 3/20 0.54
DRD4 P21917 2/20 0.54
DRD5 P21918 2/20 0.54
HTR3E A5X5Y0 1/20 0.54
MEN1 O00255 1/20 0.54
MLNR O43193 1/20 0.54
HTR3B O95264 1/20 0.54
ABCB11 O95342 1/20 0.54
ESR1 P03372 1/20 0.54
PGR P06401 1/20 0.54
ADRB2 P07550 1/20 0.54
CHRM2 P08172 1/20 0.54
ABCB1 P08183 1/20 0.54
ADRB1 P08588 1/20 0.54
HTR1A P08908 1/20 0.54
ADRA2A P08913 1/20 0.54
ADORA3 P0DMS8 1/20 0.54
GAA P10253 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23097734 0.91 GAA (0.62) DRD2HTR2ADRD3DRD5MEN1
SCHEMBL23097663 0.84 DRD2 (0.62) DRD2HTR2ADRD3DRD4HTR1A
SCHEMBL11285131 0.81 DRD2 (0.69) DRD2HTR2ASLC6A2SLC6A4HTR7
SCHEMBL23097735 0.80 GAA (0.60) DRD2HTR2ADRD3DRD4HTR1A
SCHEMBL20512952 0.79 DRD2 (1.00) DRD2
SCHEMBL30179315 0.79 DRD2 (1.00) DRD2
SCHEMBL13532793 0.79 DRD2 (0.82) DRD2HTR2ADRD3DRD4DRD5
SCHEMBL23097721 0.78 DRD2 (0.56) DRD2HTR2ADRD3DRD4HTR1A
SCHEMBL11262793 0.78 RECQL (0.66) DRD2HTR2AHTR7HRH1HRH3
SCHEMBL10665990 0.78 DRD2 (1.00) DRD2DRD3DRD4MAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118121699-A TPK agonists and methods of using the same for treating neurodegenerative diseases 上海日馨医药科技股份有限公司 2024-06-04 CN disclosed