SCHEMBL30965634

SCHEMBL30965634

O=C1CCC(Nc2ccc(N3CCC(CCN4CCC(NC(=O)OCc5ccccc5)CC4)CC3)cc2F)C(=O)N1

nearest known ligand 0.50

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CHRM4 P08173 9/20 0.50
HTR1A P08908 1/20 0.43
DRD2 P14416 1/20 0.43
HTR2A P28223 1/20 0.43
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
CHRM2 P08172 4/20 0.40
VCP P55072 1/20 0.39
CHRM5 P08912 1/20 0.37
CHRM1 P11229 1/20 0.37
CHRM3 P20309 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30965538 0.88 CHRM4 (0.45) CHRM4HTR1ADRD2HTR2AMEN1
SCHEMBL30965580 0.86 CHRM4 (0.43) CHRM4HTR1ADRD2HTR2AMEN1
SCHEMBL30965621 0.85 CHRM4 (0.39) CHRM4MEN1KMT2ACHRM2
SCHEMBL30965560 0.81 CHRM4 (0.59) CHRM4HTR1ADRD2HTR2ACHRM2
SCHEMBL30965718 0.81 CHRM4 (0.54) CHRM4HTR1ADRD2HTR2ACHRM2
SCHEMBL30965585 0.81 DDB1 (0.45) DRD2
SCHEMBL30965827 0.80 DDB1 (0.43) DRD2
SCHEMBL30136056 0.79 DDB1 (0.41) CHRM4MEN1KMT2A
SCHEMBL30965531 0.78 DDB1 (0.47) DRD2
SCHEMBL30981317 0.78 DDB1 (0.47) DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4658658-A1 NOVEL PLK1 DEGRADATION INDUCING COMPOUND Uppthera, Inc. (KR) 2025-12-10 EP disclosed
WO-2024162828-A1 NOVEL PLK1 DEGRADATION INDUCING COMPOUND UPPTHERA, INC. (KR) 2024-08-08 WO disclosed