SCHEMBL30968240

SCHEMBL30968240

N#Cc1ccnc(-c2ccc[nH]2)n1

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KDM4C Q9H3R0 1/20 0.39
CDK5 Q00535 1/20 0.37
CDK5R1 Q15078 1/20 0.37
ADORA2A P29274 1/20 0.37
ABCG2 Q9UNQ0 3/20 0.36
ABCB1 P08183 2/20 0.36
ABCC1 P33527 1/20 0.36
XDH P47989 1/20 0.35
CTSK P43235 4/20 0.35
MCL1 Q07820 1/20 0.33
NPY5R Q15761 1/20 0.33
TNKS O95271 1/20 0.31
CLK4 Q9HAZ1 1/20 0.31
MET P08581 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27920597 0.74 CDK5 (0.46) KDM4CCDK5CDK5R1ADORA2A
SCHEMBL29797941 0.74 KDM4C (0.41) KDM4CCDK5CDK5R1ABCG2ABCB1
SCHEMBL442421 0.73 KDM4C (0.46) KDM4CCDK5CDK5R1ABCG2ABCB1
SCHEMBL6131064 0.72 ABCG2 (0.53) ADORA2AABCG2ABCB1CTSKCLK4
SCHEMBL30629328 0.72 ABCG2 (0.49) ABCG2XDHCTSKMET
SCHEMBL29640777 0.69 KDM4E (0.53)
SCHEMBL31754617 0.69 KDM4E (0.53)
SCHEMBL28893597 0.68 EGLN2 (0.42) ADORA2AMCL1
SCHEMBL30968251 0.68 KDM4C (0.47) KDM4CCDK5CDK5R1
SCHEMBL13739095 0.67 TAAR1 (0.42) KDM4CCDK5CDK5R1MET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113767092-B Di-heterocyclic carbonyl substituted dihydropyrazoles, their preparation and their use in medicine 劲方医药科技(上海)有限公司 2024-07-16 CN disclosed