SCHEMBL28893597

SCHEMBL28893597

N#Cc1ccc(-c2ccc[nH]2)cn1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGLN2 Q96KS0 1/20 0.42
CHEK1 O14757 1/20 0.41
ADORA2A P29274 1/20 0.38
KDM5B Q9UGL1 1/20 0.37
VHL P40337 1/20 0.37
KDR P35968 2/20 0.37
DGAT1 O75907 1/20 0.36
TRPA1 O75762 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
RIPK1 Q13546 1/20 0.36
PDE10A Q9Y233 1/20 0.35
GABRP O00591 1/20 0.35
GABRD O14764 1/20 0.35
GABRA1 P14867 1/20 0.35
GABRB1 P18505 1/20 0.35
GABRG2 P18507 1/20 0.35
GABRB3 P28472 1/20 0.35
GABRA5 P31644 1/20 0.35
GABRA3 P34903 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12630708 0.75 CHEK1 (0.51) EGLN2CHEK1KDM5BVHLKDR
SCHEMBL30354463 0.73 HPGDS (0.53) CHEK1KDRHDAC1HDAC6IKBKE
SCHEMBL16059998 0.73 HPGDS (0.53) CHEK1KDRHDAC1HDAC6IKBKE
SCHEMBL30354464 0.73 HPGDS (0.53) CHEK1KDRHDAC1HDAC6IKBKE
SCHEMBL9215880 0.73 CYP2A6 (0.47) KDRHDAC1HDAC6PIK3CD
SCHEMBL70602 0.72 CHEK1 (0.63) EGLN2CHEK1ADORA2ADGAT1GABRP
SCHEMBL28506211 0.72 HDAC1 (0.44) ADORA2AHDAC1HDAC6RIPK1MCL1
SCHEMBL31588411 0.72 CHEK1 (0.63) EGLN2CHEK1ADORA2ADGAT1GABRP
SCHEMBL11557196 0.71 ALDH1A1 (0.60) ADORA2ARIPK1MCL1IKBKETBK1
SCHEMBL17116597 0.70 DGAT1 (0.48) EGLN2CHEK1VHLDGAT1TRPA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115368350-A PyrOX ligand containing electron-rich group at 5-position of pyridine 兰州大学 2022-11-22 CN disclosed