SCHEMBL309786

SCHEMBL309786

Cn1cc(S(=O)(=O)N(Cc2ccc(Cl)cc2)c2cccc(N3CCNC3=O)c2)cn1.O=C1NCCN1c1cccc(NCc2ccc(Cl)cc2)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 5/20 0.38
HTR2C P28335 3/20 0.37
HTR1A P08908 1/20 0.36
HTR2A P28223 1/20 0.36
HTR7 P34969 1/20 0.36
DRD3 P35462 1/20 0.36
HTR6 P50406 1/20 0.36
PKM P14618 1/20 0.35
BACE1 P56817 2/20 0.34
MEN1 O00255 3/20 0.34
KMT2A Q03164 3/20 0.34
ALDH1A1 P00352 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
LMNA P02545 2/20 0.34
POLB P06746 1/20 0.34
CNR1 P21554 4/20 0.34
NPC1 O15118 2/20 0.34
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
EGFR P00533 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3262741 0.87 KDR (0.38) HTR6BACE1MEN1KMT2ALMNA
SCHEMBL1976235 0.85 CNR2 (0.44) CNR2HTR2CHTR1AHTR2AHTR7
SCHEMBL1989680 0.85 HTR2C (0.37) CNR2HTR2CHTR1AHTR2AHTR7
SCHEMBL303078 0.80 CNR2 (0.55) CNR2HTR2CHTR1AHTR2AHTR7
SCHEMBL1966538 0.78 LMNA (0.42) HTR6BACE1MEN1KMT2ALMNA
SCHEMBL318081 0.78 DRD4 (0.39) CNR2HTR2CHTR1AHTR2AHTR7
SCHEMBL1971605 0.77 CNR2 (0.38) CNR2HTR2CHTR1AHTR2AHTR7
SCHEMBL3262739 0.73 POLB (0.47) LMNAPOLBNPC1EGFRFGFR1
SCHEMBL1965541 0.73 KMT2A (0.52) CNR2HTR2CHTR1AHTR2AHTR7
SCHEMBL302086 0.73 CNR2 (0.43) CNR2HTR2CHTR1AHTR2AHTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2012500835-A 2012-01-12 JP claimed
EP-2334637-A1 NOVEL POTASSIUM CHANNEL BLOCKERS Xention Limited (GB) 2011-06-22 EP claimed
EP-2334637-A1 NOVEL POTASSIUM CHANNEL BLOCKERS Xention Limited (GB) 2011-06-22 EP disclosed