SCHEMBL30995158

SCHEMBL30995158

CCOC(=O)Nc1cc2ccc(C#N)cc2n1C1CC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 9/20 0.43
OPRM1 P35372 1/20 0.40
OPRD1 P41143 1/20 0.40
OPRK1 P41145 1/20 0.40
OPRL1 P41146 1/20 0.40
CYP11B1 P15538 6/20 0.40
ALDH1A1 P00352 3/20 0.39
KDM4E B2RXH2 2/20 0.39
TSHR P16473 2/20 0.39
HSD17B10 Q99714 2/20 0.39
USP2 O75604 1/20 0.39
POLB P06746 1/20 0.39
HPGD P15428 1/20 0.39
ADORA2A P29274 1/20 0.38
CHRM3 P20309 2/20 0.36
CHRM2 P08172 1/20 0.36
CHRM4 P08173 1/20 0.36
CHRM5 P08912 1/20 0.36
CHRM1 P11229 1/20 0.36
SIRT2 Q8IXJ6 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30995134 0.81 CYP11B2 (0.46) CYP11B2OPRM1OPRD1OPRK1CYP11B1
SCHEMBL30995235 0.80 HSD17B10 (0.41) CYP11B2CYP11B1ALDH1A1KDM4ETSHR
SCHEMBL30995122 0.78 KMT2A (0.54) CYP11B2ALDH1A1KDM4ETSHRHSD17B10
SCHEMBL30995204 0.78 CYP11B2 (0.40) CYP11B2CYP11B1ALDH1A1ADORA2ACHRM3
SCHEMBL30995123 0.77 MAPT (0.43) CYP11B2OPRM1OPRD1OPRK1ALDH1A1
SCHEMBL30995127 0.77 HSD17B10 (0.41) CYP11B2ALDH1A1KDM4ETSHRHSD17B10
SCHEMBL21771755 0.72 KDM2B (0.36) CYP11B2CYP11B1ALDH1A1KDM4ETSHR
SCHEMBL21771753 0.72 KDM4E (0.39) CYP11B2ALDH1A1KDM4ETSHRHSD17B10
SCHEMBL21771754 0.72 KDM4E (0.39) CYP11B2ALDH1A1KDM4ETSHRHSD17B10
SCHEMBL30995226 0.71 CYP11B2 (0.53) CYP11B2CYP11B1ALDH1A1KDM4ETSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118530160-A Aromatic heterocyclic compound, preparation method and application thereof 上海翊石医药科技有限公司 2024-08-23 CN disclosed