SCHEMBL31005

SCHEMBL31005

COc1ccc(F)c(C(=O)Nc2nc3ccc(OC)cc3s2)c1

nearest known ligand 0.83

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 11/20 0.83
NPC1 O15118 10/20 0.83
KMT2A Q03164 8/20 0.71
MEN1 O00255 7/20 0.71
SCD O00767 5/20 0.71
HSD17B1 P14061 1/20 0.70
HSD17B2 P37059 1/20 0.70
SMN1; SMN2 Q16637 5/20 0.67
CYP1A2 P05177 1/20 0.67
CYP3A4 P08684 1/20 0.67
CYP2C19 P33261 1/20 0.67
HTT P42858 1/20 0.67
DYRK1A Q13627 1/20 0.67
KDM4E B2RXH2 4/20 0.67
TP53 P04637 3/20 0.67
HPGD P15428 3/20 0.67
MAPT P10636 3/20 0.67
ALDH1A1 P00352 2/20 0.67
HSD17B10 Q99714 2/20 0.67
PKM P14618 1/20 0.67

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4919731 0.91 RAB9A (1.00) RAB9ANPC1KMT2AMEN1SCD
SCHEMBL30919 0.88 RAB9A (0.72) RAB9ANPC1KMT2AMEN1SCD
SCHEMBL30930 0.87 NPC1 (0.73) RAB9ANPC1KMT2AMEN1SCD
SCHEMBL30517 0.85 RAB9A (0.82) RAB9ANPC1KMT2AMEN1SCD
SCHEMBL31001 0.84 SCD (0.76) RAB9ANPC1KMT2AMEN1SCD
SCHEMBL31087 0.84 DCLK1 (0.67) RAB9ANPC1KMT2AMEN1SCD
SCHEMBL16681363 0.84 SCD (0.88) RAB9ANPC1KMT2AMEN1SCD
SCHEMBL2480611 0.83 SCD (1.00) RAB9ANPC1KMT2AMEN1SCD
SCHEMBL10064451 0.83 SCD (1.00) RAB9ANPC1KMT2AMEN1SCD
SCHEMBL12199354 0.83 SCD (1.00) RAB9ANPC1KMT2AMEN1SCD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2609089-A1 SELECTIVE 17BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 INHIBITORS Universität des Saarlandes (DE) 2013-07-03 EP disclosed
WO-2012025638-A1 SELECTIVE 17BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 INHIBITORS Universität des Saarlandes (DE) 2012-03-01 WO disclosed
WO-2012025638-A1 SELECTIVE 17BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 INHIBITORS Universität des Saarlandes (DE) 2012-03-01 WO disclosed