SCHEMBL30517

SCHEMBL30517

COc1ccc2nc(NC(=O)c3cccc(F)c3OC)sc2c1

nearest known ligand 0.82

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 12/20 0.82
NPC1 O15118 11/20 0.82
KMT2A Q03164 8/20 0.70
MEN1 O00255 7/20 0.70
POLB P06746 1/20 0.66
SCD O00767 8/20 0.66
SMN1; SMN2 Q16637 4/20 0.63
MAPT P10636 2/20 0.63
KDM4E B2RXH2 3/20 0.61
TP53 P04637 2/20 0.61
HPGD P15428 2/20 0.61
ALDH1A1 P00352 1/20 0.61
PKM P14618 1/20 0.61
NFKB1 P19838 1/20 0.61
RECQL P46063 1/20 0.61
NFKB2 Q00653 1/20 0.61
RELA Q04206 1/20 0.61
HSD17B10 Q99714 1/20 0.61
CYP1A2 P05177 1/20 0.61
CYP3A4 P08684 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4919731 0.90 RAB9A (1.00) RAB9ANPC1KMT2AMEN1POLB
SCHEMBL31050 0.89 HSD17B1 (0.68) RAB9ANPC1KMT2AMEN1POLB
SCHEMBL30919 0.87 RAB9A (0.72) RAB9ANPC1KMT2AMEN1POLB
SCHEMBL31005 0.85 RAB9A (0.83) RAB9ANPC1KMT2AMEN1POLB
SCHEMBL30847 0.85 RAB9A (0.75) RAB9ANPC1KMT2AMEN1POLB
SCHEMBL2486652 0.83 RAB9A (0.75) RAB9ANPC1KMT2AMEN1POLB
SCHEMBL4918858 0.83 RAB9A (0.76) RAB9ANPC1KMT2AMEN1POLB
SCHEMBL4920242 0.82 RAB9A (0.79) RAB9ANPC1KMT2AMEN1POLB
SCHEMBL16562091 0.81 RAB9A (0.78) RAB9ANPC1KMT2AMEN1POLB
SCHEMBL12199352 0.81 NPC1 (0.71) RAB9ANPC1KMT2AMEN1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2609089-A1 SELECTIVE 17BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 INHIBITORS Universität des Saarlandes (DE) 2013-07-03 EP disclosed
WO-2012025638-A1 SELECTIVE 17BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 INHIBITORS Universität des Saarlandes (DE) 2012-03-01 WO disclosed
WO-2012025638-A1 SELECTIVE 17BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 INHIBITORS Universität des Saarlandes (DE) 2012-03-01 WO disclosed