SCHEMBL31033242

SCHEMBL31033242

CCOC(=O)c1cnn(Cc2cnc(N3CC4C(C3)C4(F)F)nc2C)c1

nearest known ligand 0.45

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KLKB1 P03952 13/20 0.45
POLB P06746 1/20 0.38
MAPT P10636 1/20 0.38
GRM2 Q14416 1/20 0.37
ACACB O00763 2/20 0.36
BTK Q06187 1/20 0.35
PIK3CD O00329 1/20 0.35
NR1H2 P55055 1/20 0.33
NR1H3 Q13133 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21713031 1.00 KLKB1 (0.45) KLKB1POLBMAPTGRM2ACACB
SCHEMBL21712913 0.88 KLKB1 (0.47) KLKB1BTK
SCHEMBL23469581 0.87 KLKB1 (0.56) KLKB1POLBMAPTGRM2ACACB
Lithium Ion SCHEMBL31033178 0.87 KLKB1 (0.48) KLKB1BTK
SCHEMBL21713014 0.85 KLKB1 (0.59) KLKB1
SCHEMBL30140690 0.85 KLKB1 (0.59) KLKB1
SCHEMBL20541378 0.84 KLKB1 (0.45) KLKB1POLB
SCHEMBL30140745 0.84 KLKB1 (0.45) KLKB1POLB
SCHEMBL21736734 0.83 KLKB1 (0.41) KLKB1POLBMAPTGRM2PIK3CD
SCHEMBL23769156 0.81 KLKB1 (0.51) KLKB1GRM2BTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113039181-B Heteroaromatic carboxamide derivatives as inhibitors of plasma kallikrein 勃林格殷格翰国际有限公司 2024-08-13 CN disclosed