SCHEMBL31035784

SCHEMBL31035784

CCOC(=O)c1cc2nc(C)ccn2n1

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 7/20 0.49
POLB P06746 2/20 0.49
CYP1A2 P05177 1/20 0.47
GAA P10253 3/20 0.44
MAPK1 P28482 1/20 0.44
RAB9A P51151 5/20 0.43
NPC1 O15118 3/20 0.43
RXFP1 Q9HBX9 1/20 0.43
ALDH1A1 P00352 2/20 0.43
HPGD P15428 2/20 0.43
KMT2A Q03164 4/20 0.43
L3MBTL1 Q9Y468 1/20 0.42
MAPT P10636 2/20 0.42
TSHR P16473 1/20 0.41
MEN1 O00255 1/20 0.41
THRB P10828 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23727661 0.86 KDM4E (0.47) KDM4EPOLBCYP1A2GAARAB9A
SCHEMBL21033151 0.85 KDM4E (0.48) KDM4EPOLBGAAMAPK1RAB9A
SCHEMBL23728535 0.80 APOBEC3A (0.53) KDM4EPOLBGAARAB9ANPC1
SCHEMBL4794765 0.77 APOBEC3A (0.61) KDM4EPOLBCYP1A2GAARAB9A
SCHEMBL3561838 0.76 MAPT (0.55) KDM4EPOLBCYP1A2GAAMAPK1
SCHEMBL30896072 0.74 DRD2 (0.47) KDM4EPOLBCYP1A2GAAKMT2A
SCHEMBL18343709 0.74 KDM4E (0.47) KDM4EPOLBCYP1A2GAARAB9A
SCHEMBL25887632 0.73 MAPT (0.48) KDM4EPOLBCYP1A2GAAALDH1A1
SCHEMBL18343707 0.73 KDM4E (0.46) KDM4EPOLBCYP1A2GAAMAPK1
SCHEMBL21192982 0.72 CYP1A2 (0.45) KDM4EPOLBCYP1A2GAARAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118434744-A Nitrogen-containing macrocyclic compound, and preparation method and medical application thereof 中国医药研究开发中心有限公司 2024-08-02 CN disclosed