SCHEMBL3105058

SCHEMBL3105058

CSCc1cn(C(=O)NCc2ccc(C(F)(F)F)cc2)nn1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LSS P48449 1/20 0.41
TP53 P04637 2/20 0.41
LMNA P02545 2/20 0.40
KCNH2 Q12809 1/20 0.40
HRH3 Q9Y5N1 1/20 0.40
P2RX7 Q99572 2/20 0.39
NAMPT P43490 1/20 0.39
MTOR P42345 1/20 0.39
HDAC1 Q13547 2/20 0.39
POLB P06746 1/20 0.39
HDAC3 O15379 1/20 0.39
HDAC2 Q92769 1/20 0.39
HDAC10 Q969S8 1/20 0.39
HDAC11 Q96DB2 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
PTGER4 P35408 1/20 0.39
MAPT P10636 1/20 0.38
EPHX2 P34913 1/20 0.38
PPARG P37231 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3107539 0.87 DDT (0.46) HRH3NPC1
SCHEMBL3109421 0.86 EPHX2 (0.45) HRH3NAMPTPTGER4EPHX2PPARG
SCHEMBL3113914 0.78 GLS (0.51) NAMPTEPHX2
SCHEMBL3105042 0.71 GLS (0.52) LSS
SCHEMBL17276548 0.69 KLKB1 (0.47) LSSTP53LMNAKCNH2P2RX7
SCHEMBL2629356 0.67 LSS (0.59) LSSP2RX7NAMPTMTORHDAC1
SCHEMBL24575984 0.66 MTOR (0.69) LSSNAMPTMTORHDAC1HDAC3
SCHEMBL17276449 0.66 ALDH1A1 (0.55) TP53HDAC1POLBHDAC3HDAC6
SCHEMBL12648418 0.66 ASAH1 (0.54) TP53LMNANAMPTPOLBHDAC6
SCHEMBL5464853 0.65 MEN1 (0.70) LSSKCNH2HRH3P2RX7NAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7803822-B2 Triazole derivative and use thereof TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-09-28 US disclosed