SCHEMBL31053008

SCHEMBL31053008

CC(CSc1ccnc(C(C)C)c1N)C(=O)O.COC(=O)CCSc1ccnc(CC(C)C)c1N

nearest known ligand 0.32

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.32
ALDH1A1 P00352 1/20 0.32
RAB9A P51151 1/20 0.32
KMT2A Q03164 1/20 0.32
GSTP1 P09211 1/20 0.31
GSTM2 P28161 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29238689 0.86 GSTP1 (0.38) MEN1ALDH1A1RAB9AKMT2AGSTP1
SCHEMBL22848181 0.84 GSTP1 (0.40) MEN1ALDH1A1RAB9AKMT2AGSTP1
SCHEMBL31053010 0.66 KRAS (0.35)
SCHEMBL24660012 0.65 CCNC (0.42) ALDH1A1KMT2A
SCHEMBL21852192 0.65 GSTP1 (0.42) MEN1ALDH1A1RAB9AKMT2AGSTP1
SCHEMBL21855915 0.64 CXCR1 (0.42) MEN1ALDH1A1RAB9AKMT2AGSTP1
SCHEMBL18320494 0.64 KMT2A (0.43) MEN1ALDH1A1RAB9AKMT2AGSTP1
SCHEMBL30660933 0.64 KMT2A (0.43) MEN1ALDH1A1RAB9AKMT2AGSTP1
SCHEMBL29506185 0.64 CXCR1 (0.42) MEN1ALDH1A1RAB9AKMT2AGSTP1
SCHEMBL22848251 0.64 CCNB2 (0.39) MEN1ALDH1A1RAB9AKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114008037-B Heterocyclic compounds as KRAS G12C inhibitors 广东新契生物医药科技有限公司 2024-06-21 CN disclosed