SCHEMBL31053009

SCHEMBL31053009

CC(C)c1nccc(CC(C(=O)O)C(C)(C)C)c1-n1c(=O)[nH]c(=O)c2cc(F)c(-c3c(N)cccc3Cl)nc21.CC(C)c1nccc(CCC(=O)OC(C)(C)C)c1-n1c(=O)[nH]c(=O)c2cc(F)c(-c3c(N)cccc3Cl)nc21

nearest known ligand 0.36

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KRAS P01116 20/20 0.36
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP3A5 P20815 1/20 0.32
CYP3A7 P24462 1/20 0.32
CYP2C19 P33261 1/20 0.32
CYP3A43 Q9HB55 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22848184 0.94 KRAS (0.40) KRASCYP3A4CYP2D6CYP3A5CYP3A7
SCHEMBL22848275 0.86 KRAS (0.42) KRASCYP3A4CYP2D6CYP3A5CYP3A7
SCHEMBL29614787 0.86 KRAS (0.42) KRASCYP3A4CYP2D6CYP3A5CYP3A7
SCHEMBL31052998 0.85 KRAS (0.46) KRAS
SCHEMBL22848276 0.78 KRAS (0.51) KRAS
SCHEMBL31053005 0.78 KRAS (0.35) KRAS
SCHEMBL22848337 0.72 KRAS (0.41) KRAS
SCHEMBL24436453 0.71 KRAS (0.48) KRAS
SCHEMBL29614983 0.71 KRAS (0.48) KRAS
SCHEMBL22848173 0.71 KRAS (0.47) KRAS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114008037-B Heterocyclic compounds as KRAS G12C inhibitors 广东新契生物医药科技有限公司 2024-06-21 CN disclosed