SCHEMBL31055431

SCHEMBL31055431

CC(C)(C)CNC(=O)c1ccnc(Br)c1

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 1/20 0.50
PREP P48147 1/20 0.48
CNR2 P34972 5/20 0.48
CNR1 P21554 3/20 0.48
LMNA P02545 3/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
HTT P42858 1/20 0.47
AR P10275 2/20 0.44
L3MBTL1 Q9Y468 1/20 0.43
CA12 O43570 2/20 0.42
CA9 Q16790 2/20 0.42
KDM1A O60341 1/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
NAMPT P43490 1/20 0.41
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30469331 0.86 LOXL2 (0.51) PREPLMNASMN1; SMN2HTTCA12
SCHEMBL25307043 0.82 PREP (0.45) ADORA2APREPCNR2LMNASMN1; SMN2
SCHEMBL31055445 0.80 GAA (0.59) PREPCNR2LMNASMN1; SMN2HTT
SCHEMBL3299192 0.79 HPGD (0.51) PREPHTTL3MBTL1KDM1AHDAC1
SCHEMBL3033385 0.79 HPGD (0.55) L3MBTL1NPC1KDM4EALDH1A1
SCHEMBL31055425 0.79 HTT (0.55) CNR1LMNASMN1; SMN2HTTNAMPT
SCHEMBL2998198 0.78 KDM4E (0.55) PREPLMNASMN1; SMN2HTTL3MBTL1
SCHEMBL31638112 0.78 HDAC6 (0.50) PREPSMN1; SMN2HTTARCA12
SCHEMBL8068299 0.78 ADORA2A (0.56) ADORA2ASMN1; SMN2L3MBTL1CA9NPC1
SCHEMBL30315883 0.78 KDM4E (0.55) PREPLMNASMN1; SMN2HTTL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118480001-A C-Kit (V559D)/PDGFR beta double-target allosteric inhibitor and preparation method, pharmaceutical composition and application thereof 贵州省天然产物研究中心 2024-08-13 CN disclosed