SCHEMBL31056397

SCHEMBL31056397

CC(=O)N[C@H]1CCc2cc(NC(=O)OC(C)(C)C)ccc21

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 2/20 0.52
CA1 P00915 2/20 0.52
CA9 Q16790 2/20 0.52
CA2 P00918 1/20 0.52
CA7 P43166 1/20 0.52
CA14 Q9ULX7 1/20 0.52
NPY1R P25929 1/20 0.46
TRPV1 Q8NER1 9/20 0.43
SIRT2 Q8IXJ6 3/20 0.42
SIRT1 Q96EB6 2/20 0.42
RAB9A P51151 2/20 0.41
NPC1 O15118 1/20 0.41
LMNA P02545 2/20 0.41
CYP2C9 P11712 2/20 0.41
TSHR P16473 2/20 0.41
MITF O75030 1/20 0.41
KMT2A Q03164 1/20 0.41
GMNN O75496 1/20 0.41
SLC22A3 O75751 1/20 0.41
TUBB4A P04350 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31753154 1.00 CA12 (0.52) CA12CA1CA9CA2CA7
SCHEMBL20809519 0.83 PYGL (0.47) CA12CA1CA9NPY1RSIRT2
SCHEMBL31752513 0.82 CA12 (0.59) CA12CA1CA9CA2CA7
SCHEMBL13653136 0.81 CA12 (0.45) CA12CA1CA9CA2CA7
SCHEMBL14902975 0.81 CA12 (0.45) CA12CA1CA9CA2CA7
SCHEMBL31730541 0.80 NPY1R (0.50) CA1CA2NPY1RRAB9ANPC1
SCHEMBL31055934 0.80 NPY1R (0.50) CA1CA2NPY1RRAB9ANPC1
SCHEMBL15199648 0.80 CA12 (0.43) CA12CA1CA9NPY1RSIRT2
SCHEMBL31056014 0.79 MGLL (0.51) CA12CA1CA9CA2CA7
SCHEMBL24817021 0.78 TRPV1 (0.47) CA12CA1CA9CA2CA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12570655-B2 Cysteine covalent modifiers of AKT1 and uses thereof TERREMOTO BIOSCIENCES, INC. (US) 2026-03-10 US disclosed
WO-2025081045-A9 CYSTEINE COVALENT MODIFIERS OF AKT1 AND USES THEREOF TERREMOTO BIOSCIENCES, INC. (US) 2025-12-26 WO disclosed
US-20250289819-A1 CYSTEINE COVALENT MODIFIERS OF AKT1 AND USES THEREOF TERREMOTO BIOSCIENCES, INC. 2025-09-18 US disclosed
WO-2025081045-A1 CYSTEINE COVALENT MODIFIERS OF AKT1 AND USES THEREOF TERREMOTO BIOSCIENCES, INC. (US) 2025-04-17 WO disclosed
WO-2025034613-A1 3H-IMIDAZO[4,5-B]PYRIDINE COMPOUNDS AS NON-COVALENT MODIFIERS OF AKT1 AND USES THEREOF TERREMOTO BIOSCIENCES, INC. (US) 2025-02-13 WO disclosed
WO-2024178390-A1 COVALENT MODIFIERS OF AKT1 AND USES THEREOF TERREMOTO BIOSCIENCES, INC. (US) 2024-08-29 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12570655-B2 Cysteine covalent modifiers of AKT1 and uses thereof AKT1, AKT2, AKT3 CA12 1769/4885CA1 1957/4885CA9 1752/4885
US-20250289819-A1 CYSTEINE COVALENT MODIFIERS OF AKT1 AND USES THEREOF AKT1, AKT2, AKT3 CA12 2747/4885CA1 2242/4885CA9 2779/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.