Mitoxantrone

Mitoxantrone

SCHEMBL31060880

CC(=O)O.CC(=O)O.O=C1c2c(O)ccc(O)c2C(=O)c2c(NCCNCCO)ccc(NCCNCCO)c21

nearest known ligand 0.86

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

TOP2A

The experimentally established mechanism targets of Mitoxantrone. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TOP2A known ✓ P11388 2/20 0.86
MEN1 O00255 4/20 0.86
KMT2A Q03164 4/20 0.86
BLM P54132 3/20 0.86
LMNA P02545 3/20 0.86
MAPK1 P28482 3/20 0.86
TDP1 Q9NUW8 3/20 0.86
SMN1; SMN2 Q16637 3/20 0.86
NSD2 O96028 3/20 0.86
NPC1 O15118 3/20 0.86
RAB9A P51151 3/20 0.86
USP2 O75604 2/20 0.86
TP53 P04637 2/20 0.86
RECQL P46063 2/20 0.86
MTOR P42345 2/20 0.86
CSNK2A2 P19784 2/20 0.86
CSNK2B P67870 2/20 0.86
CSNK2A1 P68400 2/20 0.86
HIF1A Q16665 2/20 0.86
CSNK2A3 Q8NEV1 2/20 0.86

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Mitoxantrone SCHEMBL31237733 1.00 MEN1 (0.86) MEN1KMT2ABLMLMNAMAPK1
Mitoxantrone SCHEMBL119801 1.00 MEN1 (0.86) MEN1KMT2ABLMLMNAMAPK1
Mitoxantrone SCHEMBL21874585 0.93 MEN1 (0.89) MEN1KMT2ABLMLMNAMAPK1
SCHEMBL11391594 0.93 MEN1 (1.00) MEN1KMT2ABLMLMNAMAPK1
Mitoxantrone SCHEMBL20214110 0.93 MEN1 (1.00) MEN1KMT2ABLMLMNAMAPK1
SCHEMBL11041207 0.93 MEN1 (1.00) MEN1KMT2ABLMLMNAMAPK1
Mitoxantrone SCHEMBL3000 0.93 MEN1 (1.00) MEN1KMT2ABLMLMNAMAPK1
SCHEMBL11517949 0.93 MEN1 (1.00) MEN1KMT2ABLMLMNAMAPK1
SCHEMBL11036806 0.93 MEN1 (1.00) MEN1KMT2ABLMLMNAMAPK1
Mitoxantrone SCHEMBL29720597 0.93 MEN1 (1.00) MEN1KMT2ABLMLMNAMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4662319-A2 PERSONALIZED CRISPR PROFILING FOR CANCER Integrate Bioscience LLC (US) 2025-12-17 EP disclosed
WO-2024168301-A2 PERSONALIZED CRISPR PROFILING FOR CANCER FUNCTION ONCOLOGY, INC. (US) 2024-08-15 WO disclosed